G. A. Weisenburger

发表

Pilot-Plant Preparation of an αvβ3 Integrin Antagonist: Process Development of a Carbonyldiimidazole Peptide Coupling

Gerald A. Weisenburger, D. Keith Anderson, Jerry D. Clark, 2009 .

Development of the Commercial Route for the Manufacture of a 5-Lipoxygenase Inhibitor PF-04191834

Shu Yu, C. Mojica, K. Leeman, 2015 .

Development of Migita Couplings for the Manufacture of a 5‐Lipoxygenase Inhibitor

Shu Yu, C. Mojica, K. Leeman, 2013 .

A comparative study of amide-bond forming reagents in aqueous media – Substrate scope and reagent compatibility

Roger M. Howard, Steven J. Fussell, Iain Robert Gladwell, 2017 .

Large-Scale Applications of Amide Coupling Reagents for the Synthesis of Pharmaceuticals

Gerald A. Weisenburger, Javier Magano, Joshua R. Dunetz, 2016 .

Dynamic thermodynamic resolution: control of enantioselectivity through diastereomeric equilibration.

M. Curtis, D. Pippel, P. Beak, 2000, Accounts of chemical research.

Solid-State Structural Investigation of an Organolithium (-)-Sparteine Complex: η3 -N-Boc-N-(p-methoxyphenyl)-3-phenylallyllithium⋅(-)-Sparteine.

D. Pippel, P. Beak, G. A. Weisenburger, 1998, Angewandte Chemie.

Ligand Control and Asymmetric Michael Reactions of Enantioenriched Configurationally Stable N-Boc Anilino Benzylic and Allylic Organolithium Species

P. Beak, Y. Park, G. A. Weisenburger, 1997 .

α-Lithiation of N-(tert-Butoxycarbonyl)-N-(p- methoxyphenyl)allylamines Mediated by (−)-Sparteine: Enantioselective Syntheses of Either Enantiomer of 3-Substituted Enecarbamates

P. Beak, G. A. Weisenburger, 1996 .

Kinetics and mechanism of the (-)-sparteine-mediated deprotonation of (E)-N-Boc-N-(p-methoxyphenyl)-3-cyclohexylallylamine.

D. Pippel, P. Beak, G. A. Weisenburger, 2001, Journal of the American Chemical Society.

Pilot Plant Preparation of an αvβ3 Integrin Antagonist. Part 1. Process Research and Development of a (S)-β-Amino Acid Ester Intermediate: Synthesis via a Scalable, Diastereoselective Imino-Reformatsky Reaction

Gerald A. Weisenburger, Thomas E. Rogers, Christine M. V. Moore, 2004 .

Festkörperstruktur des Organolithium‐(−)‐Spartein‐Komplexes η3‐N‐Boc‐N‐(p‐methoxyphenyl)‐ 3‐phenylallyllithium⋅(−)‐Spartein

D. Pippel, P. Beak, G. A. Weisenburger, 1998 .

Streamlined Synthesis of a Bicyclic Amine Moiety Using an Enzymatic Amidation and Identification of a Novel Solid Form

S. G. Ruggeri, S. Kulkarni, Amber M. Johnson, 2021 .

Determination of Reaction Heat : A Comparison of Measurement and Estimation Techniques

Ying-wei Kang, Geraldine Patricia Taber, Jerry D. Clark, 2007 .

Early Clinical Development of Lufotrelvir as a Potential Therapy for COVID-19

David W. Place, Brian P. Jones, J. Mousseau, 2023, Organic process research & development.

Temperature- and Electrophile-Dependent Stereocontrol: A Structural and Mechanistic Investigation of (−)-Sparteine-Mediated Asymmetric Lithiation−Substitution Sequences of N-Boc-N-(p-Methoxyphenyl)cinnamylamine

P. Beak, G. A. Weisenburger, N. C. Faibish, 1999 .

Practical Considerations and Examples in Adapting Amidations to Continuous Flow Processing in Early Development

Bryan Li, Gerald A. Weisenburger, James Christopher McWilliams, 2020 .

Dynamic thermodynamic resolution: control of enantioselectivity through diastereomeric equilibration.

G. A. Weisenburger, Peter Beak, David R. Anderson, 2000, Accounts of chemical research.

Synthesis of Nirmatrelvir: Development of Magnesium Sulfate-Mediated Aminolysis for the Manufacture of the Eastern Fragment

J. A. Ragan, Hatice G. Yayla, Johnny W Lee, 2023, Organic Process Research & Development.

Synthesis of Nirmatrelvir: Design and Optimization of an Efficient Telescoped Amidation–Dehydration Sequence

David W. Place, J. A. Ragan, C. Allais, 2023, Organic Process Research & Development.

Safety Notables: Information from the Literature

P. F. Vogt, G. A. Weisenburger, 2003 .