E. Mesaros

发表

BASE-INDUCED REARRANGEMENT OF O-BENZOYLBENZALDEHYDE CYANOHYDRIN TO BENZIL AND THE FURTHER REACTIONS OF BENZIL

B. Långström, G. Plé, H. Lund, 1998 .

Design, synthesis, and binding affinities of pyrrolinone-based somatostatin mimetics.

R. Hirschmann, Amos B. Smith, O. Kikuchi, 2005, Organic letters.

Discovery of Clinical Candidate CEP-37440, a Selective Inhibitor of Focal Adhesion Kinase (FAK) and Anaplastic Lymphoma Kinase (ALK).

A. Ghose, P. Dobrzanski, E. Bruckheimer, 2016, Journal of medicinal chemistry.

Synthesis and stereochemistry of some 1,3-dioxane diacetals of o-phthaldialdehyde

R. Martínez, I. Grosu, G. Plé, 1997 .

A selective, orally bioavailable 1,2,4-triazolo[1,5-a]pyridine-based inhibitor of Janus kinase 2 for use in anticancer therapy: discovery of CEP-33779.

Jennifer L. Mason, Pawel Dobrzanski, Bruce D. Dorsey, 2012, Journal of medicinal chemistry.

Stereocontrolled construction of tetrahydrofurans and gamma-butyrolactones using organomolybdenum chemistry.

A. J. Pearson, E. Mesaros, A. Pearson, 2001, Organic letters.

2,7-disubstituted-pyrrolo[2,1-f][1,2,4]triazines: new variant of an old template and application to the discovery of anaplastic lymphoma kinase (ALK) inhibitors with in vivo antitumor activity.

A. Ghose, B. Ruggeri, D. Gingrich, 2011, Journal of medicinal chemistry.

Evolution of a total synthesis of (-)-kendomycin exploiting a Petasis-Ferrier rearrangement/ring-closing olefin metathesis strategy.

E. Meyer, Amos B. Smith, E. Mesaros, 2006, Journal of the American Chemical Society.

Total synthesis of (-)-kendomycin exploiting a Petasis-Ferrier rearrangement/ring-closing olefin metathesis synthetic strategy.

E. Meyer, Amos B. Smith, E. Mesaros, 2005, Journal of the American Chemical Society.

SYNTHESIS AND STEREOCHEMISTRY OF SOME NEW 1,3-DIOXANE DERIVATIVES OF o-PHTHALDIALDEHYDE

I. Grosu, G. Plé, S. Mager, 1998 .

Study on the atropisomerism of some new 2-aryl-1,3-dioxanes

I. Grosu, G. Plé, S. Mager, 1998 .

Synthesis and stereochemistry of some dispiro-1,3-dioxanes with axial and helical chirality

I. Grosu, G. Plé, S. Mager, 1996 .

Tuberculous Lesions in Slaughter Pigs from the Viewpoint of Food Hygiene

E. Mesaros, M. Pavlas, V. Patloková, 1985 .

Discovery of VNRX-7145 (VNRX-5236 Etzadroxil): An Orally Bioavailable β-Lactamase Inhibitor for Enterobacterales Expressing Ambler Class A, C, and D Enzymes

D. Daigle, Allison L. Zulli, Bin Liu, 2021, Journal of medicinal chemistry.

Transition Metal Carbonyl Compounds

P. Serp, L. Oro, M. Ciriano, 2004 .

Piperidine-3,4-diol and piperidine-3-ol derivatives of pyrrolo[2,1-f][1,2,4]triazine as inhibitors of anaplastic lymphoma kinase.

B. Ruggeri, R. Haltiwanger, B. Dorsey, 2015, Bioorganic & medicinal chemistry letters.

Strategies to mitigate the bioactivation of 2-anilino-7-aryl-pyrrolo[2,1-f][1,2,4]triazines: identification of orally bioavailable, efficacious ALK inhibitors.

K. Wells-Knecht, H. Breslin, B. Dorsey, 2012, Journal of medicinal chemistry.

Novel 2,3,4,5-tetrahydro-benzo[d]azepine derivatives of 2,4-diaminopyrimidine, selective and orally bioavailable ALK inhibitors with antitumor efficacy in ALCL mouse models.

Andrew V. Anzalone, Jason P. Burke, B. Ruggeri, 2011, Bioorganic & medicinal chemistry letters.

Anaplastic lymphoma kinase inhibitors as anticancer therapeutics: a patent review

B. Dorsey, G. R. Ott, E. Mesaros, 2014, Expert opinion on therapeutic patents.

Methanesulfonamido-cyclohexylamine derivatives of 2,4-diaminopyrimidine as potent ALK inhibitors.

T. Underiner, B. Dorsey, T. Angeles, 2011, Bioorganic & medicinal chemistry letters.

Immunofluorescent detection of transmissible gastroenteritis virus in the intestines of piglets.

Z. Pospíšil, J. Štěpánek, E. Mesaros, 2010, Zentralblatt fur Veterinarmedizin. Reihe B. Journal of veterinary medicine. Series B.

SYNTHESIS AND STEREOCHEMISTRY OF CHIRAL 1,3-DIOXANIC COMPOUNDS OBTAINED FROM ALPHA -ALKYLATED BETA -KETOESTERS

R. Martínez, I. Grosu, G. Plé, 1995 .

2,7-Disubstituted-pyrrolotriazine kinase inhibitors with an unusually high degree of reactive metabolite formation.

M. Yazdanian, K. Wells-Knecht, D. Gingrich, 2011, Chemical research in toxicology.

Piperidine-3,4-diol and piperidine-3-ol derivatives of pyrrolo[2,1-f][1,2,4]triazine as inhibitors of anaplastic lymphoma kinase.

R. Haltiwanger, B. Dorsey, T. Angeles, 2015, Bioorganic & medicinal chemistry letters.

Diastereoselective conjugate additions to pi-allylmolybdenum complexes: a stereocontrolled route to 3,4,5-trisubstituted gamma-butyrolactones.

E. Mesaros, A. Pearson, 2002, Organic letters.

Diastereoselective Conjugate Additions to π-Allylmolybdenum Complexes: A Stereocontrolled Route to 3,4,5-Trisubstituted γ-Butyrolactones.

E. Mesaros, A. Pearson, 2010 .