K. Ekena

发表

Human estrogen receptor ligand activity inversion mutants: receptors that interpret antiestrogens as estrogens and estrogens as antiestrogens and discriminate among different antiestrogens.

B. Katzenellenbogen, M. Montano, K. Ekena, 1996, Molecular endocrinology.

Endosomolysis by masking of a membrane-active agent (EMMA) for cytoplasmic release of macromolecules.

D. L. Lewis, J. Wolff, D. Rozema, 2003, Bioconjugate chemistry.

Estrogen receptors: selective ligands, partners, and distinctive pharmacology.

B. Katzenellenbogen, J. Katzenellenbogen, M. Montano, 2000, Recent progress in hormone research.

The VPS1 protein, a homolog of dynamin required for vacuolar protein sorting in Saccharomyces cerevisiae, is a GTPase with two functionally separable domains

T. Stevens, C. Raymond, C. Vater, 1992, The Journal of cell biology.

The VPS1 protein is a dynamin-like GTPase required for sorting proteins to the yeast vacuole.

T. Stevens, C. Raymond, C. Vater, 1993, Ciba Foundation symposium.

Biologically active maleamic acid derivatives with labile amide bonds

Darren H. Wakefield, J. Hagstrom, J. Wolff, 2003 .

Constitutively active human estrogen receptors containing amino acid substitutions for tyrosine 537 in the receptor protein.

B. Katzenellenbogen, J. A. Thomas, G. Lazennec, 1996, Molecular endocrinology.

The Saccharomyces cerevisiae MVP1 gene interacts with VPS1 and is required for vacuolar protein sorting

T. Stevens, K. Ekena, 1995, Molecular and cellular biology.

Activation of a new proline transport system in Salmonella typhimurium

S. Maloy, M. Liao, K. Ekena, 1990, Journal of bacteriology.

Antiestrogens: Mechanisms of action and resistance in breast cancer

B. Katzenellenbogen, M. Montano, M. Herman, 1997, Breast Cancer Research and Treatment.

An estrogen receptor-selective coregulator that potentiates the effectiveness of antiestrogens and represses the activity of estrogens.

B. Katzenellenbogen, M. Montano, P. Martini, 1999, Proceedings of the National Academy of Sciences of the United States of America.

Determinants of Ligand Specificity of Estrogen Receptor-α: Estrogen versus Androgen Discrimination*

B. Katzenellenbogen, J. Katzenellenbogen, K. Ekena, 1998, The Journal of Biological Chemistry.

William L. McGuire Memorial Lecture. Antiestrogens: mechanisms of action and resistance in breast cancer.

B. Katzenellenbogen, M. Montano, M. Herman, 1997, Breast cancer research and treatment.

Different Residues of the Human Estrogen Receptor Are Involved in the Recognition of Structurally Diverse Estrogens and Antiestrogens*

B. Katzenellenbogen, J. Katzenellenbogen, J A Katzenellenbogen, 1997, The Journal of Biological Chemistry.

Identification of Amino Acids in the Hormone Binding Domain of the Human Estrogen Receptor Important in Estrogen Binding*

B. Katzenellenbogen, J. Katzenellenbogen, K. Weis, 1996, The Journal of Biological Chemistry.