J. Rodrigues

发表

Synthesis of 5H‐indeno[1,2‐b]pyridine derivatives: Antiproliferative and antimetastatic activities against two human prostate cancer cell lines

J. Charris, Katiuska E Charris, J. Rodrigues, 2021, Archiv der Pharmazie.

SYNTHESIS, 1H-NMR AND 13C-NMR SPECTRAL CHARACTERIZATION OF SOME ETHYL 3-AMINO-9-METHYLTHIENO[2,3-b]-4-QUINOLONE-2-CARBOXYLATES AS POTENTIAL ANTIMALARIAL AGENTS

J. Charris, J. Domínguez, J. Rodrigues, 2005 .

Potential antitumour and pro-oxidative effects of (E)-methyl 2-(7-chloroquinolin-4-ylthio)-3-(4-hydroxyphenyl) acrylate (QNACR)

F. Antunes, J. Charris, J. Rodrigues, 2013, Journal of enzyme inhibition and medicinal chemistry.

Synthesis and antimalarial activity of urenyl Bis-chalcone in vitro and in vivo

J. Domínguez, M. Acosta, J. Rodrigues, 2013, Journal of enzyme inhibition and medicinal chemistry.

Synthesis of chlorovinyl sulfones as structural analogs of chalcones and their antiplasmodial activities.

J. Gut, P. Rosenthal, J. Domínguez, 2009, European journal of medicinal chemistry.

Synthesis and evaluation of sulfonylurea derivatives as novel antimalarials.

J. Gut, P. Rosenthal, J. Charris, 2007, European journal of medicinal chemistry.

Synthesis and antimalarial activity of E-2-quinolinylbenzocycloalcanones.

J. Charris, J. Domínguez, J. Rodrigues, 2005, European journal of medicinal chemistry.

Synthesis and antimalarial activity of sulfonamide chalcone derivatives.

J. Gut, P. Rosenthal, J. Domínguez, 2005, Farmaco.

Toxicological effects of thiomersal and ethylmercury: Inhibition of the thioredoxin system and NADP(+)-dependent dehydrogenases of the pentose phosphate pathway.

A. Holmgren, Jun Lu, C. Carvalho, 2015, Toxicology and applied pharmacology.

Antimalarial Activity of Highly Coordinative Fused Heterocycles Targeting β-Hematin Crystallization

Angel H. Romero, M. Acosta, J. Rodrigues, 2022, ACS omega.

Plasmodium berghei: in vitro and in vivo activity of dequalinium.

J. Rodrigues, N. Gamboa de Domínguez, 2007, Experimental parasitology.

Synthesis and in silico ADME/Tox profiling studies of heterocyclic hybrids based on chloroquine scaffolds with potential antimalarial activity

M. Mijares, J. Charris, J. Rodrigues, 2021, Parasitology Research.

Synthesis of [(7-Chloroquinolin-4-yl)amino]chalcones: Potential Antimalarial and Anticancer Agents

K. Jung, M. Lein, C. Abramjuk, 2009 .

N′‐Formyl‐2‐(5‐nitrothiophen‐2‐yl)benzothiazole‐6‐carbohydrazide as a potential anti‐tumour agent for prostate cancer in experimental studies

B. Nitzsche, M. Höpfner, K. Jung, 2012, The Journal of pharmacy and pharmacology.

Synthesis and antimalarial activities of optically active labdane-type diterpenes

Franklin Salazar, J. Villamizar, N. Canudas, 2009, Natural product research.

Synthesis and antimalarial activity of novel chiral and achiral benzenesulfonamides bearing 1, 3, 4-oxadiazole moieties

C. Supuran, M. Zareef, J. Zaidi, 2007, Journal of enzyme inhibition and medicinal chemistry.

Synthesis, β-hematin inhibition studies and antimalarial evaluation of new dehydroxy isoquine derivatives against Plasmodium berghei: A promising antimalarial agent.

Angel H. Romero, C. Ciangherotti, S. López, 2017, European journal of medicinal chemistry.

Synthesis, crystal structure and effect of indeno[1,2-b]indole derivatives on prostate cancer in vitro. Potential effect against MMP-9.

K. Jung, M. Lein, C. Abramjuk, 2015, European journal of medicinal chemistry.

Synthesis and evaluation of new antimalarial phenylurenyl chalcone derivatives.

Jiri Gut, J. Gut, P. Rosenthal, 2005, Journal of medicinal chemistry.

Cytotoxic effects of N'-formyl-2-(5-nitrothiophen-2-yl) benzothiazole-6-carbohydrazide in human breast tumor cells by induction of oxidative stress.

F. Antunes, J. Charris, J. Rodrigues, 2012, Anticancer research.

Synthesis, antimalarial activity, structure-activity relationship analysis of thieno-[3,2-b]benzothiazine S,S-dioxide analogs.

Arthur Barazarte, S. Andujar, Daniel Enriz, 2008, Bioorganic & medicinal chemistry.

Synthesis and biological evaluation of benzimidazole-5-carbohydrazide derivatives as antimalarial, cytotoxic and antitubercular agents.

R. Gilman, R. Rojas, A. Vaisberg, 2011, Bioorganic & medicinal chemistry.

Effect of quinolinyl acrylate derivatives on prostate cancer in vitro and in vivo

B. Nitzsche, K. Jung, M. Lein, 2012, Investigational New Drugs.

Synthesis and antimalarial and anticancer evaluation of 7‐chlorquinoline‐4‐thiazoleacetic derivatives containing aryl hydrazide moieties

J. D. de Sanctis, M. Mijares, J. Charris, 2021, Archiv der Pharmazie.

Cytotoxic and apoptosis-inducing effect of ent-15-oxo-kaur-16-en-19-oic acid, a derivative of grandiflorolic acid from Espeletia schultzii.

F. Arvelo, A. Usubillaga, J. Rodrigues, 2008, Phytochemistry.

Synthesis and in silico ADME/Tox profiling studies of heterocyclic hybrids based on chloroquine scaffolds with potential antimalarial activity

M. Mijares, J. Charris, J. Rodrigues, 2021, Parasitology Research.

Synthesis and Antimalarial Activity of (E) 2-(2-Chloro-3-Quinolinylmethylidene)-5,7-Dimethoxyindanones

J. Charris, J. Domínguez, G. Lobo, 2007 .

Synthesis and biological activity of 2-[2-(7-chloroquinolin-4-ylthio)-4-methylthiazol-5-yl]-N-phenylacetamide derivatives as antimalarial and cytotoxic agents

J. D. de Sanctis, M. Mijares, J. Charris, 2020 .

Modification of oxidative status in Plasmodium berghei-infected erythrocytes by E-2-chloro-8-methyl-3-[(4'-methoxy-1'-indanoyl)-2'-methyliden]-quinoline compared to chloroquine.

J. Charris, J. Rodrigues, J. Angel, 2009, Memorias do Instituto Oswaldo Cruz.

New 4-Maleamic Acid and 4-Maleamide Peptidyl Chalcones as Potential Multitarget Drugs for Human Prostate Cancer

B. Nitzsche, M. Höpfner, C. Stephan, 2011, Pharmaceutical Research.

Antimalarial Activity of some Kaurenes

A. Usubillaga, M. Acosta, Rosa Aparicio, 2017, Natural product communications.

Synthesis and antimalarial activity of pyrazolo and pyrimido benzothiazine dioxide derivatives.

J. Charris, S. López, G. Lobo, 2009, European journal of medicinal chemistry.

Toxicological effects of thiomersal and ethylmercury: Inhibition of the thioredoxin system and NADP(+)-dependent dehydrogenases of the pentose phosphate pathway.

A. Holmgren, Jun Lu, C. Carvalho, 2015, Toxicology and applied pharmacology.

Effects of 5,8-dimethylthieno[2,3-b]quinoline-2-carboxylic acid on the antioxidative defense and lipid membranes in Plasmodium berghei-infected erythrocytes.

N. G. Domínguez, J. Rodrigues, M. Monasterios, 2015, Experimental parasitology.

Effect of dequalinium on the oxidative stress in Plasmodium berghei-infected erythrocytes

J. Rodrigues, N. Gamboa, 2009, Parasitology Research.

Modulation of the oxidative stress in malaria infection by clotrimazole

J. Rodrigues, N. Gamboa, 2012 .

Potential antitumour and pro-oxidative effects of (E)-methyl 2-(7-chloroquinolin-4-ylthio)-3-(4-hydroxyphenyl) acrylate (QNACR)

F. Antunes, J. Charris, J. Rodrigues, 2013, Journal of Enzyme Inhibition and Medicinal Chemistry.