Srinivas Olepu

发表

2-Oxo-tetrahydro-1,8-naphthyridines as selective inhibitors of malarial protein farnesyltransferase and as anti-malarials.

D. Chakrabarti, M. Gelb, C. Verlinde, 2008, Bioorganic & Medicinal Chemistry Letters.

Dialkylimidazole inhibitors of Trypanosoma cruzi sterol 14α-demethylase as anti-Chagas disease agents.

M. Gelb, F. Buckner, C. Verlinde, 2013, Bioorganic & medicinal chemistry letters.

Identification of N-[(5-{[(4-Methylphenyl)sulfonyl]amino}-3-(trifluoroacetyl)-1H-indol-1-yl)acetyl]-l-leucine (NTRC-824), a Neurotensin-like Nonpeptide Compound Selective for the Neurotensin Receptor Type 2

L. Gendron, James B. Thomas, S. Runyon, 2014, Journal of medicinal chemistry.

Second generation tetrahydroquinoline-based protein farnesyltransferase inhibitors as antimalarials.

D. Chakrabarti, M. Gelb, F. Buckner, 2007, Journal of medicinal chemistry.

The amide linker in nonpeptide neurotensin receptor ligands plays a key role in calcium signaling at the neurotensin receptor type 2.

James B. Thomas, S. Runyon, R. Wiethe, 2015, Bioorganic & medicinal chemistry letters.

Identification of N-{[6-chloro-4-(2,6-dimethoxyphenyl)quinazolin-2-yl]carbonyl}-l-leucine (NTRC-808), a novel nonpeptide chemotype selective for the neurotensin receptor type 2.

James B. Thomas, S. Runyon, R. Wiethe, 2015, Bioorganic & medicinal chemistry letters.

Identification of 1-({[1-(4-Fluorophenyl)-5-(2-methoxyphenyl)-1H-pyrazol-3-yl]carbonyl}amino)cyclohexane Carboxylic Acid as a Selective Nonpeptide Neurotensin Receptor Type 2 Compound

L. Gendron, James B. Thomas, S. Runyon, 2014, Journal of medicinal chemistry.

Structurally simple inhibitors of lanosterol 14alpha-demethylase are efficacious in a rodent model of acute Chagas disease.

M. Gelb, F. Buckner, C. Verlinde, 2009, Journal of medicinal chemistry.

5-Fluoro-2-indolyl des-chlorohalopemide (FIPI), a Phospholipase D Pharmacological Inhibitor That Alters Cell Spreading and Inhibits Chemotaxis

M. Gelb, H. Ren, G. Du, 2009, Molecular Pharmacology.

5-Fluoro-2-indolyl des-chlorohalopemide (FIPI), a Phospholipase D Pharmacological Inhibitor That Alters Cell Spreading and Inhibits Chemotaxis

M. Gelb, H. Ren, G. Du, 2009, Molecular Pharmacology.

Second generation tetrahydroquinoline-based protein farnesyltransferase inhibitors as antimalarials.

D. Chakrabarti, F. Buckner, C. Verlinde, 2007, Journal of medicinal chemistry.

2-Oxo-tetrahydro-1,8-naphthyridines as Selective Inhibitors of Malarial Protein Farnesyltransferase and as Antimalarials.

D. Chakrabarti, M. Gelb, W. V. Voorhis, 2008 .