P. Savechenkov

发表

Multiple Propofol-binding Sites in a γ-Aminobutyric Acid Type A Receptor (GABAAR) Identified Using a Photoreactive Propofol Analog*♦

R. Eckenhoff, D. C. Chiara, Jonathan B. Cohen, 2014, The Journal of Biological Chemistry.

Discovery of Tetrahydropyridopyrimidines as Irreversible Covalent Inhibitors of KRAS-G12C with In Vivo Activity.

J. Blake, J. Christensen, B. Brandhuber, 2018, ACS medicinal chemistry letters.

Identification of the Clinical Development Candidate MRTX849, a Covalent KRASG12C Inhibitor for the Treatment of Cancer

J. Blake, J. Christensen, G. Vigers, 2020 .

Anion binding modes in meso-substituted hexapyrrolic calix[4]pyrrole isomers.

P. Anzenbacher, T. Minami, Yuanli Liu, 2014, Journal of the American Chemical Society.

General Anesthetic Binding Sites in Human (cid:2) 4 (cid:3) 3 (cid:4) (cid:5) -Aminobutyric Acid Type A Receptors (GABA A Rs) *

D. C. Chiara, Jonathan B. Cohen, K. Miller, 2020 .

Allyl m-trifluoromethyldiazirine mephobarbital: an unusually potent enantioselective and photoreactive barbiturate general anesthetic.

D. Raines, D. C. Chiara, Jonathan B. Cohen, 2012, Journal of medicinal chemistry.

Anion Sensing by Fluorescent Expanded Calixpyrroles.

P. Anzenbacher, T. Minami, Ryuhei Nishiyabu, 2018, Chemistry.

Oxidation of aromatic compounds: XII. Regio- and stereoselective oxidative dimerization of alkyl 3-arylpropynoates in the system CF3CO2H-CH2Cl2-PbO2

A. Vasil’ev, P. Savechenkov, A. P. Rudenko, 2004 .

Synthesis and pharmacological evaluation of neurosteroid photoaffinity ligands.

D. C. Chiara, Jonathan B. Cohen, K. Miller, 2017, European journal of medicinal chemistry.

Protonation of 3-Arylpropynoic Acid Derivatives in Superacids

S. Walspurger, J. Sommer, P. Pale, 2005 .

Oxidation of Aromatic Compounds. Part 12. Regio- and Stereoselective Oxidation Dimerization of Alkyl 3-Arylpropynoates in the System CF3CO2H—CH2Cl2 —PbO2.

A. Vasil’ev, P. Savechenkov, A. P. Rudenko, 2005 .

Positive and Negative Allosteric Modulation of an α1β3γ2 γ-Aminobutyric Acid Type A (GABAA) Receptor by Binding to a Site in the Transmembrane Domain at the γ+-β− Interface*

D. C. Chiara, Jonathan B. Cohen, K. Miller, 2015, The Journal of Biological Chemistry.

A photoreactive analog of allopregnanolone enables identification of steroid-binding sites in a nicotinic acetylcholine receptor

D. C. Chiara, Jonathan B. Cohen, K. Bruzik, 2019, The Journal of Biological Chemistry.

Inhibitable photolabeling by neurosteroid diazirine analog in the β3-Subunit of human hetereopentameric type A GABA receptors.

D. C. Chiara, Jonathan B. Cohen, K. Miller, 2019, European journal of medicinal chemistry.

Identifying Drugs that Bind Selectively to Intersubunit General Anesthetic Sites in the α1β3γ2 GABAAR Transmembrane Domain

D. C. Chiara, Jonathan B. Cohen, K. Miller, 2019, Molecular Pharmacology.

Specificity of Intersubunit General Anesthetic-binding Sites in the Transmembrane Domain of the Human α1β3γ2 γ-Aminobutyric Acid Type A (GABAA) Receptor*♦

D. C. Chiara, Jonathan B. Cohen, K. Miller, 2013, The Journal of Biological Chemistry.

General Anesthetic Binding Sites in Human α4β3δ γ-Aminobutyric Acid Type A Receptors (GABAARs)*

D. C. Chiara, Jonathan B. Cohen, K. Miller, 2016, The Journal of Biological Chemistry.

Photoreactive Propofol Analog R ) Identified Using aA ( GABA-Aminobutyric Acid Type A Receptor γ Multiple Propofol-binding Sites in a Neurobiology :

R. Eckenhoff, D. C. Chiara, Jonathan B. Cohen, 2014 .

Binding site location on GABAA receptors determines whether mixtures of intravenous general anaesthetics interact synergistically or additively in vivo

K. Miller, K. Bruzik, P. Savechenkov, 2019, British journal of pharmacology.

p-(4-Azipentyl)propofol: a potent photoreactive general anesthetic derivative of propofol.

D. Raines, D. C. Chiara, Jonathan B. Cohen, 2011, Journal of medicinal chemistry.

Positive and Negative Allosteric Modulation of an α1β3γ2 γ-Aminobutyric Acid Type A (GABAA) Receptor by Binding to a Site in the Transmembrane Domain at the γ+-β− Interface*

D. C. Chiara, Jonathan B. Cohen, K. Miller, 2015, The Journal of Biological Chemistry.