T. Dejneka

发表

Affinity purification of endothia protease with a novel renin inhibitor SQ 32,970.

C. Free, D. Ryono, J. Norman, 1989, Biochemical and biophysical research communications.

Beta 3 agonists. Part 1: evolution from inception to BMS-194449.

R. Gregg, A. Mathur, T. Waldron, 2001, Bioorganic & medicinal chemistry letters.

Dual metalloprotease inhibitors: mercaptoacetyl-based fused heterocyclic dipeptide mimetics as inhibitors of angiotensin-converting enzyme and neutral endopeptidase.

N. Trippodo, H. Cheung, R. Misra, 1997, Journal of medicinal chemistry.

(Phosphinyloxy)acyl amino acid inhibitors of angiotensin converting enzyme (ACE). 1. Discovery of (S)-1-[6-amino-2-[[hydroxy(4-phenylbutyl)phosphinyl]oxy]-1-oxohexyl]-L -proline a novel orally active inhibitor of ACE.

D W Cushman, D. W. Cushman, J. M. Deforrest, 1988, Journal of medicinal chemistry.

(Phosphinyloxy)acyl amino acid inhibitors of angiotensin converting enzyme. 2. Terminal amino acid analogues of (S)-1-[6-amino-2 [[hydroxy(4-phenylbutyl)phosphinyl]oxy]-1-oxohexyl]-L-proline.

D W Cushman, V. Lee, D. W. Cushman, 1990, Journal of medicinal chemistry.

Aminodiol HIV protease inhibitors. Synthesis and structure-activity relationships of P1/P1' compounds: correlation between lipophilicity and cytotoxicity.

Ping Chen, S. Spergel, O. Kocy, 1996, Journal of medicinal chemistry.

A general synthesis of dioxolenone prodrug moieties

M. Poss, P. Cheng, J. Robl, 2002 .

Thyroid receptor ligands. Part 2: Thyromimetics with improved selectivity for the thyroid hormone receptor beta.

Johan Malm, Howard Einspahr, Arthur M Doweyko, 2004, Bioorganic & medicinal chemistry letters.

Quinoline-4-carboxylic acids as angiotensin II receptor antagonists

T. Waldron, S. Moreland, K. Dickinson, 1994 .

1,4-substituted indoles: a potent and selective class of angiostensin II receptor antagonists

M. Poss, Z. Gu, T. Waldron, 1994 .

BMS-201620: a selective beta 3 agonist.

T. Waldron, K. Dickinson, R. George, 2004, Bioorganic & medicinal chemistry letters.

Diol sulfonamides: A potent and novel class of inhibitors of human renin

M. Poss, T. Waldron, C. Free, 1993 .