J. Lepagnol

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Structure-activity relationships in a series of 2(1H)-quinolones bearing different acidic function in the 3-position: 6,7-dichloro-2(1H)-oxoquinoline-3-phosphonic acid, a new potent and selective AMPA/kainate antagonist with neuroprotective properties.

P. Lestage, A. Cordi, P. Morain, 1996, Journal of medicinal chemistry.

Dephosphorylation studies of SKNSH-SY 5Y cell Tau proteins by endogenous phosphatase activity

A. Delacourte, M. Caillet-Boudin, C. Soulié, 1996, Neuroscience Letters.

A new rapid method for phospholipid separation by high-performance liquid chromatography with light-scattering detection.

L. Breton, B. Serkiz, J. Volland, 1989, Journal of chromatography.

Suppression of nitric oxide formation by tyrosine kinase inhibitors in murine N9 microglia

B. Lockhart, J. Lepagnol, K. C. Cressey, 1998, British journal of pharmacology.

New Directions in Cerebral Ischemia: Sodium and Calcium Channel Modulators

M. Spedding, A. Lombet, P. Morain, 1995 .

Involvement of nicotinergic mechanisms in thyrotropin-releasing hormone-induced neurologic recovery after concussive head injury in the mouse.

P. Lestage, J. Lepagnol, A. Iris-Hugot, 1998, European journal of pharmacology.

4H-1,2,4-Pyridothiadiazine 1,1-dioxides and 2,3-dihydro-4H-1,2, 4-pyridothiadiazine 1,1-dioxides chemically related to diazoxide and cyclothiazide as powerful positive allosteric modulators of (R/S)-2-amino-3-(3-hydroxy-5-methylisoxazol-4-yl)propionic acid receptors: design, synthesis, pharmacology,

J Delarge, P Lebrun, M. Spedding, 1998, Journal of medicinal chemistry.

New prolyl endopeptidase inhibitors: in vitro and in vivo activities of azabicyclo[2.2.2]octane, azabicyclo[2.2.1]heptane, and perhydroindole derivatives.

M. Vincent, A. Benoist, G. de Nanteuil, 1996, Journal of medicinal chemistry.

PROLYL ENDOPEPTIDASE INHIBITORS : A NEW CLASS OF MEMORY ENHANCING DRUGS

G. D. Nanteuil, J. Lepagnol, B. Portevin, 1998 .

New Prolyl Endopeptidase Inhibitors: in vitro and in vivo Activities of Azabicyclo(2.2.2)octane, Azabicyclo(2.2.1)heptane, and Perhydroindole Derivatives.

M. Vincent, A. Benoist, Y. Hervé, 1996 .

Pharmacology of sodium and calcium channel modulation in neurons: implications for neuroprotection.

M. Spedding, J. Lepagnol, 1995, Biochemical Society transactions.

Structure-activity relationships in a series of 3-sulfonylamino-2-(1H)-quinolones, as new AMPA/kainate and glycine antagonists.

J. Randle, A. Cordi, P. Désos, 1995, Bioorganic & medicinal chemistry.

Allosteric potentiation by diazoxide of AMPA receptor currents and synaptic potentials.

J. Randle, J. Lepagnol, C. Biton, 1993, European journal of pharmacology.

Competitive inhibition by NBQX of kainate/AMPA receptor currents and excitatory synaptic potentials: importance of 6-nitro substitution.

J. Randle, A. Cordi, J. Lepagnol, 1992, European journal of pharmacology.

Comparative Effects of Aging Process on Phosphatidylcholine Biosynthesis Pathway: A Key Role for CTP‐Phosphocholine Cytidylyltransferase?

J. Lepagnol, V. Heidet, 1993, Annals of the New York Academy of Sciences.

Identification and characterisation of the isomers of cyclothiazide responsible for potentiating ampa current.

A. Cordi, B. Serkiz, P. Hennig, 1994 .

ENANTIOSELECTIVE SYNTHESIS OF A PYRROLO-BENZOTHIADIAZINE DERIVATIVE S 18986, A NEW AMPA RECEPTOR POSITIVE MODULATOR

A. Cordi, B. Serkiz, P. Morain, 1996 .

Quinoxaline derivatives: structure-activity relationships and physiological implications of inhibition of N-methyl-D-aspartate and non-N-methyl-D-aspartate receptor-mediated currents and synaptic potentials.

B. Lambolez, J. Randle, A. Cordi, 1992, Molecular pharmacology.

S 17092-1, A New Post-Proline Cleaving Enzyme Inhibitor: Memory Enhancing Effects and Substance P Neuromodulatory Activity

P. Lestage, D. Favale, P. Grève, 1998 .

Safety and Clinical Efficacy of S12024 in Patients with Mild to Moderate Alzheimer’s Disease

D. Guez, H. Allain, F. Mahieux, 1997 .

S 12024-2, A Cognitive Enhancer, Interacts with Nicotinic Neurotransmission

P. Lestage, M. Méen, P. Morain, 1998 .