H. R. Lagiakos

发表

In Vitro and In Vivo Inhibition of the Mycobacterium tuberculosis Phosphopantetheinyl Transferase PptT by Amidinoureas

J. Sacchettini, J. Vendôme, V. Feher, 2022, Journal of medicinal chemistry.

Thionation of amides using a solid-supported P2S5 reagent under microwave irradiation

P. Perlmutter, M. Aguilar, Ashley Walker, 2011 .

The synthesis of Fmoc-O-allyl β-serine

P. Perlmutter, M. Aguilar, H. R. Lagiakos, 2008 .

Inhibitors of histone acetyltransferases KAT6A/B induce senescence and arrest tumour growth

Nghi Nguyen, Thomas S. Peat, Olan Dolezal, 2018, Nature.

Discovery of Acylsulfonohydrazide-Derived Lysine Acetyltransferase (KAT6A) Inhibitors as Potent Senescence-Inducing Anti-Cancer Agents.

Jayme L. Dahlin, David M. Shackleford, J. Baell, 2020, Journal of medicinal chemistry.

Inhibitors of histone acetyltransferases KAT6A/B induce senescence and arrest tumour growth

A. Strasser, G. Smyth, J. Baell, 2018, Nature.

Discovery of benzoylsulfonohydrazides as potent inhibitors of the histone acetyltransferase KAT6A.

Jayme L. Dahlin, J. Baell, M. Walters, 2019, Journal of medicinal chemistry.

Discovery of a highly potent, selective, orally bioavailable inhibitor of KAT6A/B histone acetyltransferases with efficacy against KAT6A-high ER+ breast cancer.

Chin Wee Tan, Dharmesh D. Bhuva, Eric C Greenwald, 2023, Cell chemical biology.

A Computational Physics-based Approach to Predict Unbound Brain-to-Plasma Partition Coefficient, Kp,uu

Eric Therrien, Mitsunori Kato, M. Lawrenz, 2023, J. Chem. Inf. Model..