Mickael Sorge

Azaindoles as Zinc-Binding Small-Molecule Inhibitors of the JAMM Protease CSN5.

E. Altmann, U. Hassiepen, M. Renatus, 2017, Angewandte Chemie.

Optimization of the In Vivo Potency of Pyrazolopyrimidine MALT1 Protease Inhibitors by Reducing Metabolism and Increasing Potency in Whole Blood.

M. Renatus, M. Wartmann, S. Melkko, 2020, Journal of medicinal chemistry.

Stabilizing Inactive Conformations of MALT1 as an Effective Approach to Inhibit Its Protease Activity

M. Renatus, C. Wiesmann, F. Villard, 2020 .

JDQ443, a Structurally Novel, Pyrazole-Based, Covalent Inhibitor of KRASG12C for the Treatment of Solid Tumors.

N. Ostermann, R. Wilcken, S. Brachmann, 2022, Journal of medicinal chemistry.