A. S. Tong

发表

Synthesis and structure-activity relationships for tetrahydroisoquinoline-based inhibitors of Mycobacterium tuberculosis

Christopher B. Cooper, W. Denny, B. Palmer, 2020, Bioorganic & medicinal chemistry.

6-Cyano Analogues of Bedaquiline as Less Lipophilic and Potentially Safer Diarylquinolines for Tuberculosis

Christopher B. Cooper, W. Denny, B. Palmer, 2017, ACS medicinal chemistry letters.

3,5-Dialkoxypyridine analogues of bedaquiline are potent antituberculosis agents with minimal inhibition of the hERG channel

W. Denny, B. Palmer, S. Franzblau, 2019, Bioorganic & medicinal chemistry.

Synthetic Studies to Help Elucidate the Metabolism of the Preclinical Candidate TBAJ-876—A Less Toxic and More Potent Analogue of Bedaquiline

W. Denny, B. Palmer, C. Cooper, 2020, Molecules.

Synthesis and Structure–Activity Relationships for the Anti-Mycobacterial Activity of 3-Phenyl-N-(Pyridin-2-ylmethyl)Pyrazolo[1,5-a]Pyrimidin-7-Amines

Christopher B. Cooper, W. Denny, B. Palmer, 2022, Pharmaceuticals.

Variations in the C-unit of bedaquiline provides analogues with improved biology and pharmacology.

W. Denny, B. Palmer, S. Franzblau, 2019, Bioorganic & medicinal chemistry.

Synthesis and evaluation of analogues of the tuberculosis drug bedaquiline containing heterocyclic B-ring units

Christopher B. Cooper, W. Denny, B. Palmer, 2017, Bioorganic & medicinal chemistry letters.

Structure-activity relationships for unit C pyridyl analogues of the tuberculosis drug bedaquiline

Christopher B. Cooper, W. Denny, B. Palmer, 2019, Bioorganic & medicinal chemistry.

Structure-activity relationships for analogs of the tuberculosis drug bedaquiline with the naphthalene unit replaced by bicyclic heterocycles

W. Denny, B. Palmer, S. Franzblau, 2018, Bioorganic & medicinal chemistry.

Synthesis and structure-activity relationships for a new class of tetrahydronaphthalene amide inhibitors of Mycobacterium tuberculosis

Christopher B. Cooper, W. Denny, B. Palmer, 2021, European journal of medicinal chemistry.