L. Squarcialupi

发表

The 1,2,4-Triazolo[4,3-a]pyrazin-3-one as a Versatile Scaffold for the Design of Potent Adenosine Human Receptor Antagonists. Structural Investigations to Target the A2A Receptor Subtype.

A. Cavalli, G. Marucci, M. Buccioni, 2017, Journal of medicinal chemistry.

Remote control of movement disorders using a photoactive adenosine A2A receptor antagonist

F. Ciruela, K. Jacobson, J. Hernando, 2018, Journal of controlled release : official journal of the Controlled Release Society.

3-Hydroxy-1H-quinazoline-2,4-dione as a New Scaffold To Develop Potent and Selective Inhibitors of the Tumor-Associated Carbonic Anhydrases IX and XII.

C. Supuran, C. Ghelardini, A. Angeli, 2017, Journal of medicinal chemistry.

Fluorescent ligands for adenosine receptors.

S. Moro, S. Federico, G. Spalluto, 2013, Bioorganic & medicinal chemistry letters.

1,2,4‐Benzothiadiazine‐1,1‐dioxide Derivatives as Ionotropic Glutamate Receptor Ligands: Synthesis and Structure–Activity Relationships

R. Matucci, D. Catarzi, V. Colotta, 2014, Archiv der Pharmazie.

Characterization by flow cytometry of fluorescent, selective agonist probes of the A(3) adenosine receptor.

K. Jacobson, J. Auchampach, D. Tosh, 2013, Biochemical pharmacology.

4-Alkyloxyimino-cytosine nucleotides: tethering approaches to molecular probes for the P2Y6 receptor.

Kyle A. Brown, K. Jacobson, S. Costanzi, 2013, MedChemComm.

1,2,4-triazolo[1,5-a]quinoxaline derivatives and their simplified analogues as adenosine A₃ receptor antagonists. Synthesis, structure-affinity relationships and molecular modeling studies.

C. Martini, M. Betti, D. Dal Ben, 2015, Bioorganic & medicinal chemistry.

Synthesis, structure-affinity relationships, and molecular modeling studies of novel pyrazolo[3,4-c]quinoline derivatives as adenosine receptor antagonists.

K. Varani, G. Cristalli, F. Vincenzi, 2011, Bioorganic & medicinal chemistry.

The role of 5-arylalkylamino- and 5-piperazino- moieties on the 7-aminopyrazolo[4,3-d]pyrimidine core in affecting adenosine A1 and A2A receptor affinity and selectivity profiles

M. Sturlese, S. Moro, K. Varani, 2017, Journal of enzyme inhibition and medicinal chemistry.

Exploring the 2- and 5-positions of the pyrazolo[4,3-d]pyrimidin-7-amino scaffold to target human A1 and A2A adenosine receptors.

K. Varani, F. Vincenzi, M. Betti, 2016, Bioorganic & medicinal chemistry.

Exploring the 7-oxo-thiazolo[5,4-d]pyrimidine core for the design of new human adenosine A3 receptor antagonists. Synthesis, molecular modeling studies and pharmacological evaluation.

K. Varani, F. Vincenzi, M. Betti, 2015, European journal of medicinal chemistry.

7-Amino-2-phenylpyrazolo[4,3-d]pyrimidine derivatives: structural investigations at the 5-position to target human A₁ and A(2A) adenosine receptors. Molecular modeling and pharmacological studies.

S. Moro, K. Varani, F. Vincenzi, 2014, European journal of medicinal chemistry.

2-Arylpyrazolo[4,3-d]pyrimidin-7-amino derivatives as new potent and selective human A3 adenosine receptor antagonists. Molecular modeling studies and pharmacological evaluation.

S. Moro, K. Varani, C. Corciulo, 2013, Journal of medicinal chemistry.

Structural refinement of pyrazolo[4,3-d]pyrimidine derivatives to obtain highly potent and selective antagonists for the human A3 adenosine receptor.

S. Moro, K. Varani, F. Vincenzi, 2016, European journal of medicinal chemistry.

A comprehensive strategy in the development of a cyclodextrin-modified microemulsion electrokinetic chromatographic method for the assay of diclofenac and its impurities: Mixture-process variable experiments and quality by design.

S Furlanetto, S Orlandini, S. Furlanetto, 2016, Journal of chromatography. A.

3-Hydroxy-1H-quinazoline-2,4-dione derivatives as new antagonists at ionotropic glutamate receptors: molecular modeling and pharmacological studies.

S. Moro, F. Pedata, Davide Sabbadin, 2012, European journal of medicinal chemistry.

Pyrazolo[1,5-c]quinazoline derivatives and their simplified analogues as adenosine receptor antagonists: synthesis, structure-affinity relationships and molecular modeling studies.

K. Varani, G. Cristalli, F. Vincenzi, 2013, Bioorganic & medicinal chemistry.