Chu-Yi Yu

发表

Allyl 4,6-O-benzylidene-2-deoxy-2-tetrachlorophthalimido-β-d-glucopyranoside

Yan Qiao, Hong‐Yun Gao, Chu-Yi Yu, 2006 .

Methyl 3‐[(E)‐2‐(4‐bromobenzoylmethylidene)imidazolidin‐1‐yl]acrylate

Yan Qiao, Hong‐Yun Gao, Chu-Yi Yu, 2006 .

1-(4-Chlorophenyl)-2-(imidazolidin-2-ylidene)ethanone

Shengjiao Yan, Zhi-tang Huang, Chu-Yi Yu, 2006 .

1,3,4,6‐Tetra‐O‐acetyl‐2‐deoxy‐2‐tetrachlorophthalimido‐α‐d‐glucopyranoside

Yan Qiao, Hong‐Yun Gao, Chu-Yi Yu, 2006 .

Rapid detection of polyhydroxylated alkaloids in mulberry using leaf spray mass spectrometry

Z. Nie, Ning Zhang, Yafeng Li, 2013 .

A concise stereoselective synthesis of (-)-erycibelline.

S. Nakagawa, A. Kato, Xiang-Guo Hu, 2011, Organic & biomolecular chemistry.

Gem-difluoromethylated and trifluoromethylated derivatives of DMDP-related iminosugars: synthesis and glycosidase inhibition.

G. Fleet, A. Kato, Kyoko Kinami, 2016, Organic & biomolecular chemistry.

Synthesis of tetrazines from gem-difluoroalkenes under aerobic conditions at room temperature

Z. Fang, Xiang-Guo Hu, Chu-Yi Yu, 2017 .

Switchable Regioselectivity in the Opening of Aziridine by Fluoride: DFT Calculation and Synthesis of Fluorinated Piperidines

Wei-Qi Jiang, Nannan Yan, Xiang-Guo Hu, 2019 .

De Novo Synthesis of Orthogonally-Protected C2-Fluoro Digitoxoses and Cymaroses: Development and Application for the Synthesis of Fluorinated Digoxin.

Hong-Wei Chen, Xiang-Guo Hu, Ming Zhang, 2021, The Journal of organic chemistry.

3-Azidoazetidines as the first scaffolds for β-amino azetidine carboxylic acid peptidomimetics: azetidine iminosugars containing an acetamido group do not inhibit β-N-acetylhexosaminidases

M. Wormald, G. Fleet, S. Nakagawa, 2016 .

3-Fluoroazetidinecarboxylic Acids and trans,trans-3,4-Difluoroproline as Peptide Scaffolds: Inhibition of Pancreatic Cancer Cell Growth by a Fluoroazetidine Iminosugar.

M. Wormald, A. Kaji, Y. Kurashima, 2015, The Journal of organic chemistry.

trans, trans-2-C-Aryl-3,4-dihydroxypyrrolidines as potent and selective β-glucosidase inhibitors: Pharmacological chaperones for Gaucher disease.

Makiko Kise, A. Kato, Yueqing Jia, 2022, European journal of medicinal chemistry.

1‐Hydroxydiamantane

Chu-Yi Yu, Qian Li, Li-Ben Wang, 2006 .

Synthesis of Pyrrolidine Monocyclic Analogues of Pochonicine and Its Stereoisomers: Pursuit of Simplified Structures and Potent β-N-Acetylhexosaminidase Inhibition

G. Fleet, A. Kato, Yueqing Jia, 2020, Molecules.

Synthesis of eight stereoisomers of pochonicine: nanomolar inhibition of β-N-acetylhexosaminidases.

T. Nitoda, G. Fleet, Jian-She Zhu, 2013, The Journal of organic chemistry.

Synthesis of 2-acetamido-1,2-dideoxy-d-galacto-nojirimycin [DGJNAc] from d-glucuronolactone: the first sub-micromolar inhibitor of α-N-acetylgalactosaminidases

Andreas F. G. Glawar, T. Butters, G. Fleet, 2010 .

Total Synthesis of Pseudouridimycin.

Chu-Yi Yu, Yi-Xian Li, Xu-kun Wang, 2022, Organic letters.

First total synthesis of (+)-broussonetine W: glycosidase inhibition of natural product & analogs.

G. Fleet, A. Kato, Kyoko Kinami, 2016, Organic & biomolecular chemistry.

Facile Aerobic Alkylation of Rhodium Porphyrins with Alkyl Halides

K. Chan, Kai‐En Hung, Wu Yang, 2015 .

Rhodium-catalyzed oxidative homologation of N-pyrimidyl indolines with alkynes via dual C H activation: Facile synthesis of benzo[g]indolines

Lianhui Wang, Xiuling Cui, Dan Xiong, 2018, Chinese Chemical Letters.

Inhibition of nonmammalian glycosidases by azetidine iminosugars derived from stable 3,5-di-O-triflates of pentoses.

G. Fleet, S. Nakagawa, A. Kato, 2011, Organic letters.

Synthesis of bis‐ketene N,S‐acetals with a polymethylene linkage

Zhi-tang Huang, Chu-Yi Yu, Li-Ben Wang, 1996 .

Diastereoselective Synthesis, Glycosidase Inhibition, and Docking Study of C-7-Fluorinated Casuarine and Australine Derivatives.

Makiko Kise, G. Fleet, A. Kato, 2022, The Journal of organic chemistry.

Fluorinated Radicamine A and B: Synthesis and Glycosidase Inhibition

Xuan-Hui Zhao, M. Xiao, G. Fleet, 2016 .

Fluorinated and Conformationally Fixed Derivatives of L-HomoDMDP: Synthesis and Glycosidase Inhibition.

M. Xiao, G. Fleet, A. Kato, 2015, The Journal of organic chemistry.

Synthesis and glycosidase inhibition of australine and its fluorinated derivatives.

Wei Zhang, M. Xiao, G. Fleet, 2015, Organic letters.

Iminosugars as therapeutic agents: recent advances and promising trends.

G. Fleet, A. Kato, R. Nash, 2011, Future medicinal chemistry.

L-DMDP, L-homoDMDP and their C-3 fluorinated derivatives: synthesis and glycosidase-inhibition.

G. Fleet, A. Kato, Y. Yamashita, 2011, Organic & biomolecular chemistry.

A direct retro-Reformatsky fragmentation: formal ring enlargement of cyclic ketones for novel and practical synthesis of heterocyclic enamines.

Mei-Xin Zhao, G. Fleet, Zhi-tang Huang, 2004, The Journal of organic chemistry.

Construction of effective receptor for recognition of avian influenza H5N1 protein HA1 by assembly of monohead glycolipids on polydiacetylene vesicle surface.

Long Jiang, Long Jiang, Mingxing Duan, 2009, Bioconjugate chemistry.

Synthesis and glycosidase inhibition of N-substituted derivatives of 1,4-dideoxy-1,4-imino-d-mannitol (DIM).

G. Fleet, A. Kato, Yueqing Jia, 2020, Organic & biomolecular chemistry.

Epimerization of C5 of an N-hydroxypyrrolidine in the synthesis of swainsonine related iminosugars.

G. Fleet, A. Kato, Kyoko Kinami, 2016, Organic & biomolecular chemistry.

A novel one-pot reaction of heterocyclic ketene aminals: Synthesis of a small library of tetrahydropyridinone-fused 1,3-diazaheterocycles

Mei-Xin Zhao, Peng-Hui Yang, Zhi-tang Huang, 2006 .

Reactions of Heterocyclic Ketene Aminals with Dimethyl Oxalate: A Facile Synthesis of γ-Lactam Fused 1,3-Diazaheterocycles

Zhi-tang Huang, Chu-Yi Yu, Li-Ben Wang, 1996 .

Azetidine iminosugars from the cyclization of 3,5-di-O-triflates of α-furanosides and of 2,4-di-O-triflates of β-pyranosides derived from glucose.

R. Martínez, G. Fleet, A. Kato, 2012, Organic letters.

[1-(2-Hydroxyethyl)imidazolidin-2-ylidene]malononitrile

Yan Qiao, Hong‐Yun Gao, Chu-Yi Yu, 2006 .

Synthesis of fused N-heterocycles utilizing the heterocyclic enamine protocol

Y. Liu, Meining Wang, Chu-Yi Yu, 2003 .

Ring-chain tautomerism in organic synthesis: synthesis of heterocyclic enamines from a novel and practical formal ring transformation reaction of lactones.

Y. Liu, Hongjun Gao, Meining Wang, 2003, The Journal of organic chemistry.

Design and Synthesis of Labystegines, Hybrid Iminosugars from LAB and Calystegine, as Inhibitors of Intestinal α-Glucosidases: Binding Conformation and Interaction for ntSI.

S. Hirono, I. Nakagome, Yutaro Tsuji, 2015, The Journal of organic chemistry.

General Intermediates for the Synthesis of 6-C-Alkylated DMDP-Related Natural Products

Yueqing Jia, Chu-Yi Yu, Yi-Xian Li, 2013, Molecules.

Synthesis of fully substituted polyhydroxylated pyrrolizidines via Cope-House cyclization.

Wei Zhang, G. Fleet, A. Kato, 2011, Organic letters.

Concise synthesis of 1-epi-castanospermine

Bin Cheng, Yueqing Jia, Chu-Yi Yu, 2017 .

A concise synthesis of homochiral sedamines and related alkaloids. A new reductive application of Jacobsen's catalyst

O. Meth–Cohn, Chu-Yi Yu, 1999 .

Reactions of Heterocyclic Ketene Aminals with Baylis-Hillman Acetates : A Novel Synthesis of Tetrahydropyridine-Fused 1,3-Diazaheterocycles

M. Yaqub, Yueqing Jia, Zhi-tang Huang, 2008 .

Novel 2-aryl-3;4;5-trihydroxypiperidines: Synthesis and glycosidase inhibition

H Zhao, G. Fleet, S. Nakagawa, 2013 .

An Efficient Synthesis of Aldohexose-Derived Piperidine Nitrones: Precursors of Piperidine Iminosugars

H Zhao, Jian-She Zhu, Yueqing Jia, 2013, Molecules.

Concise synthesis of calystegines B2 and B3via intramolecular Nozaki-Hiyama-Kishi reaction.

G. Fleet, A. Kato, Kyoko Kinami, 2016, Organic & biomolecular chemistry.

Looking glass inhibitors: L-DMDP, a more potent and specific inhibitor of alpha-glucosidases than the enantiomeric natural product DMDP.

R. Dwek, M. Wormald, T. Butters, 2004, Chemical communications.

1,4-Dideoxy-2,3-O-isopropylidene-N-[3-(3-nitrobenzoylamino)benzoyl]-1,4-imino-D-talitol

Ying Fu, Chu-Yi Yu, 2006 .

Radicamines A and B: synthesis and revision of the absolute configuration.

Chu-Yi Yu, Mu-Hua Huang, 2006, Organic letters.

NHC-mediated cross-coupling of sugar-derived cyclic nitrones with enals: general and efficient synthesis of polyhydroxylated pyrrolizidines and indolizidines.

Wei Zhang, Wenqing Xu, A. Kato, 2013, Organic & biomolecular chemistry.

Synthesis and glycosidase inhibition of the enantiomer of (-)-steviamine, the first example of a new class of indolizidine alkaloid.

G. Fleet, S. Nakagawa, A. Kato, 2010, Organic letters.

Steviamine, a new indolizidine alkaloid from Stevia Rebaudiana

A. Michalik, G. Fleet, A. Kato, 2010 .

Steviamine, a new class of indolizidine alkaloid [(1R,2S,3R,5R,8aR)-3-hydroxymethyl-5-methyloctahydroindolizine-1,2-diol hydrobromide]

D. Watkin, A. Michalik, G. Fleet, 2009, Acta crystallographica. Section E, Structure reports online.

Synthesis and Glycosidase Inhibition of Broussonetine M and Its Analogues

G. Fleet, A. Kato, Kyoko Kinami, 2019, Molecules.

Design, synthesis and glycosidase inhibition of C-4 branched LAB and DAB derivatives.

Makiko Kise, G. Fleet, A. Kato, 2022, European journal of medicinal chemistry.

General synthesis of sugar-derived azepane nitrones: precursors of azepane iminosugars.

K. Izumori, G. Fleet, S. Nakagawa, 2013, The Journal of organic chemistry.

Total synthesis and glycosidase inhibition of broussonetine I and J(2).

A. Kato, Yueqing Jia, Chu-Yi Yu, 2013, The Journal of organic chemistry.

5-C-Branched Deoxynojirimycin: Strategy for Designing a 1-Deoxynojirimycin-Based Pharmacological Chaperone with a Nanomolar Affinity for Pompe Disease.

I. Nakagome, Tomoki Yoshida, N. Tanaka, 2022, Journal of medicinal chemistry.

Synthesis of a novel C-branched polyhydroxylated cyclic nitrone

Yueqing Jia, Chu-Yi Yu, Yi-Xian Li, 2017 .

Synthesis and glycosidase inhibition of C-7 modified casuarine derivatives

Bin Cheng, A. Kato, Yueqing Jia, 2017 .

Synthesis of Spiro Heterocyclic Ketene Aminals

Zhi-tang Huang, Chu-Yi Yu, Li-Ben Wang, 1996 .

Interaction of spiro[(2R,3R,4S)-4-benzyloxy-2,3-iso-propylidenedioxy-1-oxacyclopentane-5,5′-(2-nitromethylene-1,3-diazacyclohexane)] with bovine serum albumin

Yalin Tang, Jiangpeng Liao, J. Xiang, 2008 .

Synthesis and Glycosidase Inhibition of the Enantiomer of (‐)‐Steviamine, the First Example of a New Class of Indolizidine Alkaloid.

G. Fleet, S. Nakagawa, A. Kato, 2010 .

Nine of 16 stereoisomeric polyhydroxylated proline amides are potent β-N-acetylhexosaminidase inhibitors.

Andreas F. G. Glawar, M. Wormald, T. Butters, 2014, The Journal of organic chemistry.

New Synthetic Methodology en route to Asymmetric Piperidine Alkaloids

O. Meth–Cohn, Chu-Yi Yu, Cze Chak Yau, 1999 .

The Regiospecific N-Alkylation of Heterocyclic Ketene Aminals with Ethyl Bromoacetate: A Facile Route to 3-Pyrrolidinone Fused Diazaheterocycles

Zhi-tang Huang, Chu-Yi Yu, Li-Ben Wang, 1994 .

Nanomolar β-glucosidase and β-galactosidase inhibition by enantiomeric α-1-C-alkyl-1,4-dideoxy-1,4-imino-arabinitol derivatives.

Makiko Kise, G. Fleet, Tian-Tian Lu, 2022, European journal of medicinal chemistry.

Synthesis and glycosidase inhibition of N-substituted derivatives of 1,4-dideoxy-1,4-imino-d-mannitol (DIM).

G. Fleet, A. Kato, Yueqing Jia, 2020, Organic & biomolecular chemistry.

C-6 fluorinated casuarines as highly potent and selective amyloglucosidase inhibitors: Synthesis and structure-activity relationship study.

Makiko Kise, G. Fleet, A. Kato, 2022, European journal of medicinal chemistry.

A practical synthesis of sugar-derived cyclic nitrones: powerful synthons for the synthesis of iminosugars

Wei Zhang, Weihua Xu, Yueqing Jia, 2010 .