Keisuke Aihara

发表

Application of N-C- or C-N-directed sequential native chemical ligation to the preparation of CXCL14 analogs and their biological evaluation.

T. Hara, A. Otaka, Kohei Sato, 2011, Bioorganic & medicinal chemistry.

Liquid-phase synthesis of bridged peptides using olefin metathesis of a protected peptide with a long aliphatic chain anchor.

A. Otaka, Akira Shigenaga, D. Takahashi, 2015, Organic letters.

Cysteine-Free Intramolecular Ligation of N-Sulfanylethylanilide Peptide Using 4-Mercaptobenzylphosphonic Acid: Synthesis of Cyclic Peptide Trichamide

Fei-xue Fu, D. Hutchins, A. Otaka, 2017 .

A Recyclable Hydrophobic Anchor‐Tagged Asymmetric Amino Thiourea Catalyst

A. Otaka, Akira Shigenaga, Ken‐ichi Yamada, 2018, ChemCatChem.

One-Pot/Sequential Native Chemical Ligation Using Photocaged Crypto-thioester.

A. Otaka, Akira Shigenaga, T. Inokuma, 2016, Organic letters.

The total chemical synthesis of the monoglycosylated GM2 ganglioside activator using a novel cysteine surrogate.

A. Otaka, Kohei Sato, D. Tsuji, 2015, Chemical communications.

Identification of SNAIL1 Peptide-Based Irreversible Lysine-Specific Demethylase 1-Selective Inactivators.

P. Zhan, Yukihiro Itoh, Miki Suzuki, 2016, Journal of medicinal chemistry.

Stapled BIG3 helical peptide ERAP potentiates anti-tumour activity for breast cancer therapeutics

T. Katagiri, Y. Miyoshi, S. Toyokuni, 2017, Scientific Reports.

Development of an Intein-Inspired Amide Cleavage Chemical Device.

A. Otaka, Akira Shigenaga, T. Inokuma, 2016, The Journal of organic chemistry.

Synthesis of lactam-bridged cyclic peptides using sequential olefin metathesis and diimide reduction reactions

A. Otaka, Akira Shigenaga, T. Inokuma, 2015 .