Haiyan Tao

发表

Small molecule antagonists in distinct binding modes inhibit drug-resistant mutant of smoothened.

P. Schultz, Yan Wang, J. Kelleher, 2011, Chemistry & biology.

Ternary complex of human RORγ ligand‐binding domain, inverse agonist and SMRT peptide shows a unique mechanism of corepressor recruitment

R. Babine, Shin‐ichi Hirashima, Makoto Shiozaki, 2017, Genes to cells : devoted to molecular & cellular mechanisms.

Ternary crystal structure of human RORγ ligand-binding-domain, an inhibitor and corepressor peptide provides a new insight into corepressor interaction

Shin‐ichi Hirashima, Makoto Shiozaki, P. Crowe, 2018, Scientific Reports.

Discovery of Second Generation RORγ Inhibitors Composed of an Azole Scaffold.

Takayoshi Suzuki, Hiromasa Hashimoto, Makoto Shiozaki, 2019, Journal of medicinal chemistry.

Characterization of a New Glycosynthase Cloned by Using Chemical Complementation

V. Cornish, P. Peralta-Yahya, John D. Decatur, 2008, Chembiochem : a European journal of chemical biology.

Synthesis and biological evaluation of novel 2-(2-arylmethylene)hydrazinyl-4-aminoquinazoline derivatives as potent antitumor agents.

X. Zhai, Nan Jiang, P. Gong, 2012, European journal of medicinal chemistry.

Synthesis and Biological Evaluation of 4‐Phenoxy‐6,7‐disubstituted Quinolines Possessing Semicarbazone Scaffolds as Selective c‐Met Inhibitors

Di Wu, P. Gong, Jinying Bai, 2013, Archiv der Pharmazie.

A genomic screen identifies TYRO3 as a MITF regulator in melanoma

Buu P. Tu, A. Orth, L. Miraglia, 2009, Proceedings of the National Academy of Sciences.

Identification of RING finger protein 4 (RNF4) as a modulator of DNA demethylation through a functional genomics screen

A. Orth, L. Miraglia, P. Schultz, 2010, Proceedings of the National Academy of Sciences.

Milestones in directed enzyme evolution.

Virginia W Cornish, V. Cornish, Haiyan Tao, 2002, Current opinion in chemical biology.

SAR Exploration Guided by LE and Fsp(3): Discovery of a Selective and Orally Efficacious RORγ Inhibitor.

R. Babine, Shin‐ichi Hirashima, Hiromasa Hashimoto, 2016, ACS medicinal chemistry letters.

Optimized design and synthesis of chemical dimerizer substrates for detection of glycosynthase activity via chemical complementation.

Hening Lin, Virginia W Cornish, Pamela Peralta-Yahya, 2006, Bioorganic & medicinal chemistry.

Macamide B suppresses lung cancer progression potentially via the ATM signaling pathway

Yihui Xu, Haiyan Tao, Min Wang, 2023, Oncology letters.

Directed evolution of a glycosynthase via chemical complementation.

Hening Lin, Virginia W Cornish, V. Cornish, 2004, Journal of the American Chemical Society.

Clinical significance of LARGE1 in progression of liver cancer and the underlying mechanism.

Ping Huang, Min Wang, Haiyan Tao, 2021, Gene.

High-throughput selection for cellulase catalysts using chemical complementation.

Brian T. Carter, V. Cornish, Hening Lin, 2008, Journal of the American Chemical Society.