H. Falls

发表

Optimization of 2,4-diaminopyrimidines as GHS-R antagonists: side chain exploration.

H. Sham, C. Collins, Gang Liu, 2006, Bioorganic & medicinal chemistry letters.

Characterization of ghrelin receptor activity in a rat pituitary cell line RC-4B/C.

C. Collins, B. Dayton, W. Kaszubska, 2006, Journal of molecular endocrinology.

Discovery and pharmacological evaluation of growth hormone secretagogue receptor antagonists.

E. Bush, H. Sham, D. Beno, 2006, Journal of medicinal chemistry.

2,4-diaminopyrimidine derivatives as potent growth hormone secretagogue receptor antagonists.

E. Bush, H. Sham, D. Beno, 2006, Journal of medicinal chemistry.

Structure-activity relationship studies on tetralin carboxamide growth hormone secretagogue receptor antagonists.

Jyoti R. Patel, H. Sham, C. Collins, 2005, Bioorganic & medicinal chemistry letters.

Discovery of tetralin carboxamide growth hormone secretagogue receptor antagonists via scaffold manipulation.

H. Sham, C. Collins, Gang Liu, 2004, Journal of medicinal chemistry.

Novel isoxazole carboxamides as growth hormone secretagogue receptor (GHS-R) antagonists.

H. Sham, C. Collins, Gang Liu, 2004, Bioorganic & medicinal chemistry letters.

Nonsteroidal selective glucocorticoid modulators: the effect of C-10 substitution on receptor selectivity and functional potency of 5-allyl-2,5-dihydro-2,2,4-trimethyl-1H-[1]benzopyrano[3,4-f]quinolines.

S. Elmore, M. Nakane, J. Miner, 2003, Journal of medicinal chemistry.

Protein tyrosine phosphatase 1B negatively regulates leptin signaling in a hypothalamic cell line

D. White, D. Haasch, P. Kroeger, 2002, Molecular and Cellular Endocrinology.

Identification of diamino chromone-2-carboxamides as MCHr1 antagonists with minimal hERG channel activity.

G. Gintant, A. Souers, G. Diaz, 2007, Bioorganic & medicinal chemistry letters.

Identification and preliminary characterization of a potent, safe, and orally efficacious inhibitor of acyl-CoA:diacylglycerol acyltransferase 1.

Steven C. Cullen, P. Hajduk, A. Souers, 2012, Journal of medicinal chemistry.