Liwei Han

发表

N1-Substituted Quinoxaline-2,3-diones as Kainate Receptor Antagonists: X-ray Crystallography, Structure-Affinity Relationships, and in Vitro Pharmacology.

J. Kastrup, D. Pickering, K. Frydenvang, 2019, ACS chemical neuroscience.

Chemoenzymatic synthesis of new 2,4-syn-functionalized (S)-glutamate analogues and structure-activity relationship studies at ionotropic glutamate receptors and excitatory amino acid transporters.

J. Kastrup, M. Gajhede, T. Gefflaut, 2013, Journal of medicinal chemistry.

Neto2 Influences on Kainate Receptor Pharmacology and Function.

J. Howe, D. Pickering, Liwei Han, 2016, Basic & clinical pharmacology & toxicology.

Augmentation of Anticancer Drug Efficacy in Murine Hepatocellular Carcinoma Cells by a Peripherally Acting Competitive N-Methyl-d-aspartate (NMDA) Receptor Antagonist.

K. Hansen, L. Bunch, T. Malm, 2017, Journal of medicinal chemistry.

Design, synthesis and in vitro pharmacology of GluK1 and GluK3 antagonists. Studies towards the design of subtype-selective antagonists through 2-carboxyethyl-phenylalanines with substituents interacting with non-conserved residues in the GluK binding sites.

L. Olsen, D. Pickering, J. Kristensen, 2014, Bioorganic & medicinal chemistry.

Binding mode of an α-amino acid-linked quinoxaline-2,3-dione analogue at glutamate receptor subtype GluK1.

J. Kastrup, L. Bunch, D. Bowie, 2015, ACS chemical neuroscience.

( S)-2-Amino-3-(5-methyl-3-hydroxyisoxazol-4-yl)propanoic Acid (AMPA) and Kainate Receptor Ligands: Further Exploration of Bioisosteric Replacements and Structural and Biological Investigation.

Simone Brogi, Ettore Novellino, Mikko Gynther, 2018, Journal of medicinal chemistry.

Testosterone-independent down-regulation of Oct2 in the kidney medulla from a uranyl nitrate-induced rat model of acute renal failure: effects on distribution of a model organic cation, tetraethylammonium.

Dae-Duk Kim, W. Shim, C. Shim, 2009, Journal of pharmaceutical sciences.

Structure − Activity Relationship Study of Ionotropic Glutamate Receptor Antagonist ( 2 S , 3 R ) ‐ 3-( 3-Carboxyphenyl ) pyrrolidine-2-carboxylic Acid

J. Kastrup, L. Bunch, D. Pickering, 2015 .

Design and Synthesis of a Series of l-trans-4-Substituted Prolines as Selective Antagonists for the Ionotropic Glutamate Receptors Including Functional and X-ray Crystallographic Studies of New Subtype Selective Kainic Acid Receptor Subtype 1 (GluK1) Antagonist (2S,4R)-4-(2-Carboxyphenoxy)pyrrolidin

J. Kastrup, L. Bunch, D. Bowie, 2017, Journal of medicinal chemistry.

Preparation and evaluation of andrographolide-loaded microemulsion

X. Niu, Xue-zhi Yang, Hong Du, 2012, Journal of microencapsulation.

Dose dependency in the oral bioavailability of an organic cation model, tributylmethyl ammonium (TBuMA), in rats: association with the saturation of efflux by the P-gp system on the apical membrane of the intestinal epithelium.

Dae-Duk Kim, C. Shim, Yong-Hae Han, 2005, Journal of pharmaceutical sciences.

Structurally improved reduced graphene oxide nanocluster structured assembly with Naringin for the effective photothermal therapy of colon tumour patients and nursing care management

Tianyu Meng, Yuhang Wang, Juan Tan, 2020, Molecular Physics.

Decreased secretory transport of a quarternary ammonium, TBuMA, across LLC-PK1 cells by the anionic kidney extract

Dae-Duk Kim, W. Shim, C. Shim, 2008, Archives of pharmacal research.