Keletso Maepa

Lapatinib, Nilotinib and Lomitapide Inhibit Haemozoin Formation in Malaria Parasites

T. Egan, Jill M Combrinck, A. C. C. de Sousa, 2020, Molecules.

Virtual screening as a tool to discover new β-haematin inhibitors with activity against malaria parasites

T. Egan, Jill M Combrinck, A. C. C. de Sousa, 2020, Scientific Reports.

Structure-activity relationship studies of antiplasmodial cyclometallated ruthenium(II), rhodium(III) and iridium(III) complexes of 2-phenylbenzimidazoles.

K. Chibale, Dale Taylor, Gregory S. Smith, 2019, European journal of medicinal chemistry.

Identification of 2,4-Disubstituted Imidazopyridines as Hemozoin Formation Inhibitors with Fast-Killing Kinetics and In Vivo Efficacy in the Plasmodium falciparum NSG Mouse Model.

K. Chibale, T. Egan, Dale Taylor, 2020, Journal of medicinal chemistry.

THC shows activity against cultured Plasmodium falciparum.

T. Egan, Jill M Combrinck, A. C. C. de Sousa, 2021, Bioorganic & medicinal chemistry letters.

A Diverse Range of Hemozoin Inhibiting Scaffolds Act on Plasmodium falciparum as Heme Complexes.

T. Egan, Jill M Combrinck, R. Hunter, 2021, ACS infectious diseases.

Virtual screening as a tool to discover new β-haematin inhibitors with activity against malaria parasites

T. Egan, Jill M Combrinck, A. C. C. de Sousa, 2020, Scientific Reports.