C. Simeon

Novel immunomodulator FTY720 is phosphorylated in rats and humans to form a single stereoisomer. Identification, chemical proof, and biological characterization of the biologically active species and its enantiomer.

E. Francotte, M. Zollinger, V. Brinkmann, 2005, Journal of medicinal chemistry.

Direct synthesis of [DOTA-DPhe1]-octreotide and [DOTA-DPhe1,Tyr3]-octreotide (SMT487): two conjugates for systemic delivery of radiotherapeutical nuclides to somatostatin receptor positive tumors in man.

P. Smith-Jones, C. Bruns, R. Albert, 1998, Bioorganic & medicinal chemistry letters.

Medicinal chemistry of somatostatin analogs leading to the DTPA and DOTA conjugates of the multi-receptor-ligand SOM230.

D. Hoyer, R. Kneuer, C. Bruns, 2005, Journal of Endocrinological Investigation.