T. Jack

发表

Benzofuran based non-peptide antagonists of angiotensin II related to GR117289: part IV; imidazopyridinylbenzofurans.

G. Currie, A. W. Dean, D. Gallacher, 1994 .

Aryl aminopyrazole benzamides as oral non-steroidal selective glucocorticoid receptor agonists.

H. T. Jones, James M. Woolven, I. McLay, 2009, Bioorganic & medicinal chemistry letters.

Sialidase inhibitors related to zanamivir. Further SAR studies of 4-amino-4H-pyran-2-carboxylic acid-6-propylamides.

P. Colman, J. Varghese, A. Wonacott, 2001, Bioorganic & medicinal chemistry letters.

Thalidomide-based TNF-inhibitors for neurodegenerative diseases

Rogers, N. Greig, Qian-sheng Yu, 2004 .

Efficient synthesis of an α-trifluoromethyl-α-tosyloxymethyl epoxide enabling stepwise double functionalisation to afford CF3-substituted tertiary alcohols

H. T. Jones, G. Hardy, D. Coe, 2008 .

Bromobenzofuran-based non-peptide antagonists of angiotensin II: GR138950, a potent antihypertensive agent with high oral bioavailability.

D. Scopes, D. Judd, M. Dowle, 1994, Journal of medicinal chemistry.

Structure-based optimisation of orally active & reversible MetAP-2 inhibitors maintaining a tight 'molecular budget'.

P. Thomas, Jonathan D Goodacre, Lena Shukla, 2020, Bioorganic & medicinal chemistry letters.

Discovery of a potent series of non-steroidal non α-trifluoromethyl carbinol glucocorticoid receptor agonists with reduced lipophilicity.

I. McLay, Hawa Diallo, I. Uings, 2011, Bioorganic & medicinal chemistry letters.

Bromobenzofurans : a new class of potent, non-peptide antagonists of angiotensin II

J. Montana, K. Clark, M. J. Robertson, 1991 .

Benzofuran based angiotensin II antagonists related to GR117289: enhancement of potency in vitro and oral activity

J. Montana, K. Clark, M. J. Robertson, 1993 .