V. Gregor

发表

A Practical and Scalable Synthesis of GTx-134, an IGF-1R Inhibitor

Yahu A. Liu, V. Gregor, 2016 .

Optimization of alkylidene hydrazide based human glucagon receptor antagonists. Discovery of the highly potent and orally available 3-cyano-4-hydroxybenzoic acid [1-(2,3,5,6-tetramethylbenzyl)-1H-indol-4-ylmethylene]hydrazide.

A. Kuki, Michael D. Johnson, D. Murphy, 2002, Journal of medicinal chemistry.

Human glucagon receptor antagonists based on alkylidene hydrazides.

A. Kuki, D. Murphy, A. Polinsky, 2002, Bioorganic & medicinal chemistry letters.

Identification of alkylidene hydrazides as glucagon receptor antagonists.

A. Kuki, D. Murphy, A. Polinsky, 2001, Journal of medicinal chemistry.

CI‐1002: A Combined Acetylcholinesterase Inhibitor and Muscarinic Antagonist 1

C. J. Moore, M. Emmerling, J. Scholten, 1995 .

Structure-activity studies on benzhydrol-containing nipecotic acid and guvacine derivatives as potent, orally-active inhibitors of GABA uptake.

M. R. Pavia, R. Schwarz, D. Mayhugh, 1992, Journal of medicinal chemistry.

Synthesis of fluorine-18 labeled GABA uptake inhibitors.

M. Kilbourn, M. R. Pavia, V. Gregor, 1990, International journal of radiation applications and instrumentation. Part A, Applied radiation and isotopes.

Synthesis and metabolic profile of Cl‐966: A potent, orally‐active inhibitor of GABA uptake

T. Woolf, M. R. Pavia, S. Bjorge, 1990 .

Novel parallel synthesis of N-(4-oxo-2-substituted-4H-quinazolin-3-yl)-substituted sulfonamides

Yuefen Zhou, D. Murphy, Zhongxiang Sun, 2004 .

Synthesis and SAR of 3,5-diamino-piperidine derivatives: novel antibacterial translation inhibitors as aminoglycoside mimetics.

Thomas Hermann, Sarah Fish, T. Hermann, 2007, Bioorganic & medicinal chemistry letters.

ACETYLCHOLINESTERASE INHIBITION BY FUSED DIHYDROQUINAZOLINE COMPOUNDS

M. Emmerling, J. Jaén, Robert E Davis, 1996 .

Novel Parallel Synthesis of N‐(4‐Oxo‐2‐Substituted‐4H‐quinazolin‐3‐yl)‐Substituted Sulfonamides.

Yuefen Zhou, D. Murphy, Zhongxiang Sun, 2005 .

Structure-Guided Discovery of Novel Aminoglycoside Mimetics as Antibacterial Translation Inhibitors

Thomas Hermann, Sarah Fish, T. Hermann, 2005, Antimicrobial Agents and Chemotherapy.

CI-1002, a Novel Anticholinesterase and Muscarinic Antagonist

C. J. Moore, M. Emmerling, J. Scholten, 1995 .

The synthesis and in vitro acetylcholinesterase and butyrylcholinesterase inhibitory activity of tacrine (Cognex®) derivaties

C. J. Moore, M. Emmerling, V. Gregor, 1992 .

In Vitro and In Vivo Effects of a Dual Inhibitor of Acetylcholinesterase and Muscarinic Receptors, CI-1002

C. J. Moore, M. Emmerling, J. Scholten, 1994 .

PD 142676 (CI 1002), a novel anticholinesterase and muscarinic antagonist

C. J. Moore, M. Emmerling, J. Scholten, 1994, Molecular Neurobiology.