Y. Bi

发表

Tandem optimization of target activity and elimination of mutagenic potential in a potent series of N-aryl bicyclic hydantoin-based selective androgen receptor modulators.

L. Hamann, A. Fura, R. Seethala, 2007, Bioorganic & medicinal chemistry letters.

Design, synthesis, and evaluation of phenylglycinols and phenyl amines as agonists of GPR88.

Alan G. E. Wilson, Vijay T. Ahuja, Y. Liu, 2015, Bioorganic & medicinal chemistry letters.

The discovery of potent agonists for GPR88, an orphan GPCR, for the potential treatment of CNS disorders.

Y. Liu, A. Cacace, J. Macor, 2015, Bioorganic & medicinal chemistry letters.

Quinolines as extremely potent and selective PDE5 inhibitors as potential agents for treatment of erectile dysfunction.

J. Macor, J. Krupinski, A. Watson, 2004, Bioorganic & Medicinal Chemistry Letters.

The discovery of novel, potent and selective PDE5 inhibitors.

J. Macor, J. Krupinski, A. Watson, 2001, Bioorganic & medicinal chemistry letters.

Stereospecificity in the Pictet-Spengler reaction. Enantiospecific synthesis of (6S,10S)-5#75)-5-methyl-9-oxo-12-benzyl-6,7,8,9,10,11-hexahydro-6,10-imino-5H-cyclooct[b]indole, a template for preparation of macroline/sarpagine alkaloids

J. Cook, Y. Bi, Fuda Yu, 1992 .

Pharmacological and x-ray structural characterization of a novel selective androgen receptor modulator: potent hyperanabolic stimulation of skeletal muscle with hypostimulation of prostate in rats.

Stanley R Krystek, Jacek Ostrowski, K. Kish, 2007, Endocrinology.

The Solid - Phase Synthesis of Oligoureas

P. Schultz, S. Paikoff, Y. Bi, 1996 .

General approach for the synthesis of macroline/sarpagine alkaloids. The total synthesis of (+)-macroline

J. Cook, Y. Bi, 1993 .

Inhibition of AAK1 Kinase as a Novel Therapeutic Approach to Treat Neuropathic Pain

Alan G. E. Wilson, G. Shankar, S. Mandlekar, 2016, The Journal of Pharmacology and Experimental Therapeutics.

Building blocks for peptide and carbamate libraries

P. Schultz, Y. Bi, 1996 .

Checkpoint inhibition through small molecule-induced internalization of programmed death-ligand 1

Bhavna S. Paratala, R. Rijnbrand, M. Sofia, 2021, Nature Communications.

Synthesis and SAR of tetrahydropyrrolo[1,2-b][1,2,5]thiadiazol-2(3H)-one 1,1-dioxide analogues as highly potent selective androgen receptor modulators.

L. Hamann, R. Seethala, G. Grover, 2007, Bioorganic & medicinal chemistry letters.

Enantiospecific Synthesis of (-)-Alstonerine and (+)-Macroline as Well as a Partial Synthesis of (+)-Villalstonine

J. Cook, Linda K. Hamaker, Y. Bi, 1994 .

Inhibition of AAK 1 Kinase as a Novel Therapeutic Approach to Treat Neuropathic Pain s

Alan G. E. Wilson, Malley, G. Shankar, 2016 .

Design, synthesis, and evaluation of phenylglycinols and phenyl amines as agonists of GPR88.

Alan G. E. Wilson, Vijay T. Ahuja, Y. Liu, 2015, Bioorganic & medicinal chemistry letters.