J. Weatherhead

发表

Discovery of a potent boronic acid derived inhibitor of the HCV RNA-dependent RNA polymerase.

R. Hamatake, Z. Hong, Shawn P. Williams, 2014, Journal of medicinal chemistry.

Carbamoyl pyridone HIV-1 integrase inhibitors. 2. Bi- and tricyclic derivatives result in superior antiviral and pharmacokinetic profiles.

E. Garvey, T. Seki, T. Fujiwara, 2013, Journal of medicinal chemistry.

The use of oxadiazole and triazole substituted naphthyridines as HIV-1 integrase inhibitors. Part 1: Establishing the pharmacophore.

E. Garvey, S. Foster, J. Jeffrey, 2009, Bioorganic & medicinal chemistry letters.

1,3,4-Oxadiazole substituted naphthyridines as HIV-1 integrase inhibitors. Part 2: SAR of the C5 position.

E. Garvey, S. Foster, J. Jeffrey, 2009, Bioorganic & medicinal chemistry letters.

Naphthyridinone (NTD) integrase inhibitors 4. Investigating N1 acetamide substituent effects with C3 amide groups.

E. Garvey, S. Foster, T. Fujiwara, 2014, Bioorganic & medicinal chemistry letters.

Naphthyridinone (NTD) integrase inhibitors: N1 protio and methyl combination substituent effects with C3 amide groups.

E. Garvey, S. Foster, T. Fujiwara, 2013, Bioorganic & medicinal chemistry letters.

Combining symmetry elements results in potent naphthyridinone (NTD) HIV-1 integrase inhibitors.

E. Garvey, S. Foster, T. Fujiwara, 2011, Bioorganic & medicinal chemistry letters.

Pharmacovirological Impact of an Integrase Inhibitor on Human Immunodeficiency Virus Type 1 cDNA Species In Vivo

Steven J. Novick, E. Garvey, K. Chiswell, 2009, Journal of Virology.

Pharmacovirological Impact of an Integrase Inhibitor on Human Immunodeﬁciency Virus Type 1 cDNA Species In Vivo (cid:1)

Steven J. Novick, E. Garvey, K. Chiswell, 2009 .

The Naphthyridinone GSK364735 Is a Novel, Potent Human Immunodeficiency Virus Type 1 Integrase Inhibitor and Antiretroviral

E. Garvey, S. Foster, T. Fujiwara, 2007, Antimicrobial Agents and Chemotherapy.

Synthesis and pharmacokinetic profile of highly deuterated brecanavir analogs.

T. Baughman, B. Johns, D. Temelkoff, 2013, European journal of medicinal chemistry.

Pyrazolopyrimidines and pyrazolotriazines with potent activity against herpesviruses.

K. Gudmundsson, B. Johns, J. Weatherhead, 2009, Bioorganic & medicinal chemistry letters.

Carbamoyl pyridone HIV-1 integrase inhibitors 3. A diastereomeric approach to chiral nonracemic tricyclic ring systems and the discovery of dolutegravir (S/GSK1349572) and (S/GSK1265744).

E. Garvey, T. Seki, S. Foster, 2013, Journal of medicinal chemistry.