T. Boos

发表

Synthesis, radiosynthesis and in vivo evaluation of [I]-4-(2-(bis(4-fluorophenyl)methoxy)ethyl)-1-(4-iodobenzyl)piperidine as a selective tracer for imaging the dopamine transporter.

K. Rice, F. de Vos, L. Wyffels, 2009, Journal of labelled compounds & radiopharmaceuticals.

Structure-activity relationships of substituted N-benzyl piperidines in the GBR series: Synthesis of 4-(2-(bis(4-fluorophenyl)methoxy)ethyl)-1-(2-trifluoromethylbenzyl)piperidine, an allosteric modulator of the serotonin transporter.

K. Rice, R. Rothman, C. Dersch, 2006, Bioorganic & medicinal chemistry.

Studies of the Biogenic Amine Transporters. XI. Identification of a 1-[2-[Bis(4-fluorophenyl)methoxy]ethyl]-4-(3-phenylpropyl)piperazine (GBR12909) Analog That Allosterically Modulates the Serotonin Transporter

K. Rice, R. Rothman, C. Dersch, 2005, Journal of Pharmacology and Experimental Therapeutics.

3-O-Formyl-20R,21-epoxyresibufogenin suppresses IL-6-type cytokine actions by targeting the glycoprotein 130 subunit: potential clinical implications.

G. Chrousos, T. Kino, K. Rice, 2007, The Journal of allergy and clinical immunology.

An Improved Synthesis of 3β-Acetoxy-lanost-8-en-24-one (24-Ketolanosteryl Acetate)

E. Parish, S. A. Kizito, T. Boos, 2000 .

Design and synthesis of promiscuous high-affinity monoamine transporter ligands: unraveling transporter selectivity.

K. Rice, R. Rothman, C. Dersch, 2006, Journal of medicinal chemistry.

Remote functionalization of the steroid side-chain

E. Parish, Nida Aksara, T. Boos, 1997, Lipids.

Remote Functionalization of the Cholestane Side-chain by Chromyl Acetates

E. Kaneshiro, E. Parish, Nida Aksara, 1999 .

DAT/SERT selectivity of flexible GBR 12909 analogs modeled using 3D-QSAR methods.

K. Rice, R. Rothman, C. Dersch, 2007, Bioorganic & medicinal chemistry.

The Chemistry of Waxes and Sterols

E. Parish, T. L. Boos, Shengrong Li, 2002 .

In vivo evaluation of [123I]-4-(2-(bis(4-fluorophenyl)methoxy)ethyl)-1-(4-iodobenzyl)piperidine, an iodinated SPECT tracer for imaging the P-gp transporter.

Steven Staelens, Filip De Vos, Steven Deleye, 2010, Nuclear medicine and biology.

Reversal of pancreatitis-induced pain by an orally available, small molecule interleukin-6 receptor antagonist

J. Deschamps, K. Rice, F. Porreca, 2010, PAIN®.

Studies of the Biogenic Amine Transporters. XI. Identification of a 1-[2-[Bis(4-fluorophenyl)methoxy]ethyl]-4-(3-phenylpropyl)piperazine (GBR12909) Analog That Allosterically Modulates the Serotonin Transporter

K. Rice, R. Rothman, C. Dersch, 2005, Journal of Pharmacology and Experimental Therapeutics.