R. Morales

发表

Human prorenin structure sheds light on a novel mechanism of its autoinhibition and on its non-proteolytic activation by the (pro)renin receptor.

Z. Böcskei, Y. Watier, R. Morales, 2012, Journal of molecular biology.

Nanomolar inhibitors of Mycobacterium tuberculosis glutamine synthetase 1: synthesis, biological evaluation and X-ray crystallographic studies.

B. Scheiper, S. Silve, A. Bauer, 2015, Bioorganic & medicinal chemistry letters.

Structural basis for substrate selectivity and nucleophilic substitution mechanisms in human adenine phosphoribosyltransferase catalyzed reaction

B. Daignan-Fornier, R. Barouki, I. Ceballos-Picot, 2019, The Journal of Biological Chemistry.

Sensitivity of Oncogenic KRAS-Expressing Cells to CDK9 Inhibition

M. Yi, J. Frappier, F. McCormick, 2021, SLAS discovery : advancing life sciences R & D.

Crystal structures of novel non-peptidic, non-zinc chelating inhibitors bound to MMP-12.

Sophie Perrier, S. Dufour, Renaud Morales, 2004, Journal of molecular biology.

Conformational changes induced by nucleotide binding in Cdc6/ORC from Aeropyrum pernix.

Ian Grainge, N. Cook, D. Wigley, 2004, Journal of molecular biology.

Structural Insights into the Forward and Reverse Enzymatic Reactions in Human Adenine Phosphoribosyltransferase.

B. Daignan-Fornier, R. Barouki, I. Ceballos-Picot, 2018, Cell chemical biology.

Structure-based design and synthesis of novel non-zinc chelating MMP-12 inhibitors.

J. Hamon, P. Ducrot, P. Cluzeau, 2005, Bioorganic & medicinal chemistry letters.

Preparation and optimization of new 4-(morpholin-4-yl)-(6-oxo-1,6-dihydropyrimidin-2-yl)amide derivatives as PI3Kβ inhibitors.

J. Nicolas, C. Lengauer, L. Vincent, 2012, Bioorganic & medicinal chemistry letters.

Structure-based design and synthesis of novel non-zinc chelating MMP-12 inhibitors.

Pierre Ducrot, Jacques Hamon, Alexis Denis, 2005, Bioorganic & medicinal chemistry letters.