Tsuyoshi Arita

发表

Substituents at the naphthalene C3 position of (-)-Cercosporamide derivatives significantly affect the maximal efficacy as PPARγ partial agonists.

K. Wakabayashi, Shinko Hayashi, J. Ohsumi, 2012, Bioorganic & medicinal chemistry letters.

(-)-Cercosporamide derivatives as novel antihyperglycemic agents.

J. Ohsumi, K. Araki, S. Satoh, 2009, Bioorganic & medicinal chemistry letters.

Synthetic studies on apoptolidin: synthesis of the C1–C21 macrolide fragment

K. Toshima, S. Matsumura, Koji Kato, 2001 .

Discovery of a novel selective PPARgamma modulator from (-)-Cercosporamide derivatives.

K. Wakabayashi, Shinko Hayashi, J. Ohsumi, 2010, Bioorganic & medicinal chemistry letters.

Synthesis and biological evaluation of novel chiral diazepine derivatives as bombesin receptor subtype-3 (BRS-3) agonists incorporating an antedrug approach.

Y. Nagai, Yasuyuki Abe, K. Shimada, 2015, Bioorganic & medicinal chemistry.

Discovery of novel chiral diazepines as bombesin receptor subtype-3 (BRS-3) agonists with low brain penetration.

K. Shimada, Kazuhiro Yoshida, Hisashi Takahashi, 2014, Bioorganic & medicinal chemistry letters.

Discovery of a novel bicyclic compound, DS54360155, as an orally potent analgesic without mu-opioid receptor agonist activity.

K. Shimada, Nobuo Machinaga, Y. Domon, 2019, Bioorganic & medicinal chemistry letters.

Discovery of conolidine derivative DS39201083 as a potent novel analgesic without mu opioid agonist activity.

K. Shimada, Nobuo Machinaga, Y. Domon, 2019, Bioorganic & medicinal chemistry letters.

Synthesis and biological evaluation of novel (-)-Cercosporamide derivatives as potent selective PPARγ modulators.

K. Wakabayashi, Shinko Hayashi, J. Ohsumi, 2012, European journal of medicinal chemistry.

Vacuolar-type H(+)-ATPase inhibitory activity of synthetic analogues of the concanamycins: is the hydrogen bond network involving the lactone carbonyl, the hemiacetal hydroxy group, and the C-19 hydroxy group essential for the biological activity of the concanamycins?

M. Imoto, M. Ueda, Y. Yoshimoto, 2002, Bioorganic & medicinal chemistry letters.

(-)-Cercosporamide derivatives as novel antihyperglycemic agents.

J. Ohsumi, K. Araki, S. Satoh, 2009, Bioorganic & medicinal chemistry letters.