O. Pineau

The discovery of equipotent PPARalpha/gamma dual activators.

D. Grillot, Paul Martres, A. Laroze, 2008, Bioorganic & medicinal chemistry letters.

Design, synthesis and evaluation of trifluoromethane sulfonamide derivatives as new potent and selective peroxisome proliferator-activated receptor alpha agonists.

D. Grillot, Paul Martres, A. Laroze, 2008, Bioorganic & medicinal chemistry letters.

Discovery of novel indazole derivatives as dual angiotensin II antagonists and partial PPARγ agonists.

D. Grillot, E. Nicodème, Yann Lamotte, 2014, Bioorganic & medicinal chemistry letters.

Substituted 2-[(4-aminomethyl)phenoxy]-2-methylpropionic acid PPARalpha agonists. 1. Discovery of a novel series of potent HDLc raising agents.

M. Lambert, H. Xu, D. Grillot, 2007, Journal of medicinal chemistry.

Discovery of epigenetic regulator I-BET762: lead optimization to afford a clinical candidate inhibitor of the BET bromodomains.

P. Bamborough, R. Prinjha, C. Chung, 2013, Journal of medicinal chemistry.