D. Gala

发表

Mono N-arylation of piperazine(III): metal-catalyzed N-arylation and its application to the novel preparations of the antifungal posaconazole and its advanced intermediate

M. Hepperle, C. A. Evans, Lan Shen, 2002 .

An Intramolecular Silyl Transfer from the Carboxylate to the Hydroxyl Group in Sodium 4-Hydroxybutyrate and Its Application to the Synthesis of Injectable Antifungal Posaconazole Derivative, Sch 59884

B. Pramanik, Lan Shen, G. Chen, 2002 .

A rational approach to chiral α-hydroxy aryl ketones from chiral aryl epoxides via regioselective, stereo retentive oxidative epoxide opening: Its application to the synthesis of antifungal Sch 42427/SM 9164

D. Gala, D. DiBenedetto, 1994 .

Preparation of Guanine PDE Inhibitors: Development of the Common Synthetic Route Strategy. A Case Study

G. Gloor, A. Miller, D. Gala, 2004 .

A novel synthesis of guanine PDE inhibitors via tricyclic imidazopyrimidines

D. Gala, M. B. Mitchell, D. DiBenedetto, 2003 .

Tetrahydropyran as an efficient alcohol protecting group for the synthesis of penems: synthesis of Sch 34343

D. Gala, M. Steinman, R. Jaret, 1986 .

Synthesis of 8-amino-6-methoxycinnoline. A precursor for 2-azaprimaquine

R. A. Coburn, D. Gala, 1982 .

Reaction of aziridinium ions with organometallic reagents: optimization of the key step of ecopipam synthesis

I. Zavialov, V. Dahanukar, D. Gala, 2002 .

A convenient, improved synthesis of (camphoryl)sulfonyl oxaziridines.

I. Mergelsberg, D. Gala, D. DiBenedetto, 1992 .

Total chiral synthesis of azole antifungals via α-hydroxylation of ketones

I. Mergelsberg, D. Gala, M. Kugelman, 1996 .

Antitumor Imidazotetrazines. 35. New Synthetic Routes to the Antitumor Drug Temozolomide.

M. Stevens, W. Thomson, Yongfeng Wang, 1997, The Journal of organic chemistry.

Sequential mono-N-arylation of piperazine nitrogens. Part 1: A simplified method and its application to the preparation of a key N,N′-biaryl piperazine antifungal intermediate

M. Hepperle, D. Gala, M. EckertJeffrey, 1999 .

Sequential mono-N-arylation of piperazine nitrogens. Part 2: The role of hydrogen bonding

J. B. Lambert, T. Chan, D. Gala, 1999 .

Preparations of antifungal Sch 42427/SM 9164: Preparative chromatographic resolution, and total asymmetric synthesis via enzymatic preparation of chiral α-hydroxy arylketones

D. Gala, M. Steinman, D. Schumacher, 1996 .

An efficient syntesis of 1,8-naphthyridin-2(1H)-ones : synthesis of leukotriene inhibitor SCH 37224

D. Gala, M. Steinman, P. Nyce, 1991 .

Effects of the affinity ligands 14-β-chloroacetylnaltrexone and 14-β-bromoacetamidomorphine on [3H]-dihydromorphine binding sites in rat brain

M. Reichman, R. Dirksen, L. Abood, 1986 .

A novel acyclic addition of ketenes to oxazoles/oxazolines

M. Puar, D. Gala, R. Jaret, 1987 .

One-Step Synthesis of Biphenylacetic Acids via Pd/C-Catalyzed Arylation

A. Stamford, D. Gala, M. Kugelman, 1997 .

(+)-(2R, 8AR*)-(8,8-DIMETHOXYCAMPHORYL)SULFONYLOXAZIRIDINE AND (+)-(2R, 8AR*)-(8,8-DICHLOROCAMPHORYL)-SULFONYLOXAZIRIDINE : (4H-4A, 7-METHANOOXAZIRINO 3,2-I2,1BENZISOTHIAZOLE, TETRAHYDRO-8,8-DIMETHOXY-9,9-DIMETHYL-, 3,3-DIOXID E, 2R-(2ALPHA , 4AALPHA , 7ALPHA , 8AR*)- AND 4H-4A, 7-METHANOOXAZIRINO3,

Anil Kumar, P. Zhou, F. A. Davis, 1996 .

Derives de guanine 2-benzyle-polycyclique et procede de preparation

D. Gala, M. Kugelman, D. DiBenedetto, 1994 .

Guanine hydrolysis under basic conditions to substituted imidazoles

M. Czarniecki, P. Das, M. Puar, 2000 .

(+)‐(2R,8aR*)‐[(8,8‐Dimethoxycamphoryl)Sulfonyl]Oxaziridine and (+)‐(2R,8aR*)‐[(8,8‐Dichlorocamphoryl)Sulfonyl]Oxaziridine

Anil Kumar, P. Zhou, F. A. Davis, 2003 .

Metal salts induced improved α-hydroxylation of ketones for the preparation of the key chiral intermediate of azole antifungals

D. Gala, D. DiBenedetto, 1997 .

A practical conversion of an azetidinone to penem: Synthesis of Sch 34343

V. Girijavallabhan, A. Ganguly, S. McCombie, 1992 .

A Practical Conversion of an Azetidinone to Penem: Synthesis of Sch 34343.

V. Girijavallabhan, A. Ganguly, S. McCombie, 1992 .

Exploratory Process Development of a High-Temperature Thermal (3 + 2) Cycloaddition in Continuous Flow for the Synthesis of Seltorexant

L. Moens, Kiran Matcha, D. Depré, 2023, Organic Process Research & Development.

Diastereoisomerism in 1,3,5-triazine through nitrogen substituents

M. Puar, D. Gala, M. Steinman, 1994 .