S. Sagawa

发表

Discovery of 6-phenylpyrimido[4,5-b][1,4]oxazines as potent and selective acyl CoA:diacylglycerol acyltransferase 1 (DGAT1) inhibitors with in vivo efficacy in rodents.

Masahiro Tanaka, Kexue Li, Masahiro Suzuki, 2014, Journal of medicinal chemistry.

Synthesis of Anilino‐monoindolylmaleimides as Potent and Selective PKCβ Inhibitors.

Masahiro Tanaka, T. Sasase, I. Matsuda, 2005 .

Discovery of pyrrolopyridazines as novel DGAT1 inhibitors.

Masahiro Tanaka, Kexue Li, B. Shan, 2010, Bioorganic & medicinal chemistry letters.

Synthesis, SAR studies, and pharmacological evaluation of 3-anilino-4-(3-indolyl) maleimides with conformationally restricted structure as orally bioavailable PKCbeta-selective inhibitors.

Masahiro Tanaka, T. Sasase, Nobuhisa Ueda, 2006, Bioorganic & medicinal chemistry.

Catalytic Asymmetric Aminolysis of 3,5,8-Trioxabicyclo[5.1.0]octane Providing an Optically Pure 2-Amino-1,3,4-butanetriol Equivalent.

Y. Hase, T. Inaba, S. Sagawa, 1999, The Journal of organic chemistry.

Efficient synthesis of enantiomerically pure 5,5-Dimethyl-4-hydroxy-2-cyclopentenone

H. Miyaoka, S. Sagawa, H. Nagaoka, 1995 .

Novel protein kinase C‐β isoform selective inhibitor JTT‐010 ameliorates both hyper‐ and hypoalgesia in streptozotocin‐ induced diabetic rats

T. Sasase, T. Abe, M. Matsushita, 2005, Diabetes, obesity & metabolism.

EFFICIENT SYNTHESIS OF OPTICALLY ACTIVE CYCLOHEXENONES

H. Miyaoka, S. Sagawa, H. Nagaoka, 1994 .

Efficient Synthesis of Optically Active Cyclohexenones.

H. Miyaoka, S. Sagawa, H. Nagaoka, 1994 .

(1S)-1-[(4R)-2,2-dimethyl-1,3-dioxolan+-4-yl][-2-hydroxyethylamm onium benzoate, a versatile building block for chiral 2-aminoalkanols: concise synthesis and application to nelfinavir, a potent HIV-protease inhibitor.

Y. Yamada, T. Inaba, S. Sagawa, 2000, The Journal of organic chemistry.

Synthesis of anilino-monoindolylmaleimides as potent and selective PKCbeta inhibitors.

Takashi Inaba, Jun-ichi Hoshi, Tomohiko Sasase, 2004, Bioorganic & medicinal chemistry letters.