Salahuddin Mirza

发表

Sulfated Polysaccharides from Macroalgae Are Potent Dual Inhibitors of Human ATP-Hydrolyzing Ectonucleotidases NPP1 and CD39

C. Müller, J. Sévigny, J. Pelletier, 2021, Marine drugs.

Protein kinase inhibitor ceritinib blocks ectonucleotidase CD39 – a promising target for cancer immunotherapy

J. Sévigny, J. Pelletier, E. Tolosa, 2022, Journal for ImmunoTherapy of Cancer.

Targeting the Main Protease of SARS‐CoV‐2: From the Establishment of High Throughput Screening to the Design of Tailored Inhibitors

A. Schiedel, C. Müller, M. Gütschow, 2021, Angewandte Chemie.

2‐Substituted thienotetrahydropyridine derivatives: Allosteric ectonucleotidase inhibitors

M. Gütschow, J. Sévigny, J. Pelletier, 2021, Archiv der Pharmazie.

Adenine-(methoxy)-ethoxy-Pα,α-dithio-triphosphate inhibits pathologic calcium pyrophosphate deposition in osteoarthritic human chondrocytes.

C. Müller, J. Sévigny, J. Pelletier, 2019, Organic & biomolecular chemistry.

Discovery of potent nucleotide pyrophosphatase/phosphodiesterase3 (NPP3) inhibitors with ancillary carbonic anhydrase inhibition for cancer (immuno)therapy.

C. Müller, C. Supuran, N. Boshta, 2021, RSC medicinal chemistry.

Identification of adenine-N9-(methoxy)ethyl-β-bisphosphonate as NPP1 inhibitor attenuates NPPase activity in human osteoarthritic chondrocytes

J. Sévigny, J. Pelletier, B. Fischer, 2019, Purinergic Signalling.

Identification of adenine-N9-(methoxy)ethyl-β-bisphosphonate as NPP1 inhibitor attenuates NPPase activity in human osteoarthritic chondrocytes

C. Müller, J. Sévigny, J. Pelletier, 2019, Purinergic Signalling.

Synthesis and structure-activity relationships of ticlopidine derivatives and analogs as inhibitors of ectonucleotidase CD39.

J. Sévigny, J. Pelletier, Thanigaimalai Pillaiyar, 2023, Bioorganic chemistry.

Nucleotide Analog ARL67156 as a Lead Structure for the Development of CD39 and Dual CD39/CD73 Ectonucleotidase Inhibitors

C. Müller, J. Sévigny, J. Pelletier, 2020, Frontiers in Pharmacology.

Development of a selective and highly sensitive fluorescence assay for nucleoside triphosphate diphosphohydrolase1 (NTPDase1, CD39).

C. Müller, J. Sévigny, H. Stephan, 2018, The Analyst.

Heparins are potent inhibitors of ectonucleotide pyrophosphatase/phospho-diesterase-1 (NPP1) – a promising target for the immunotherapy of cancer

J. Pelletier, G. Bendas, O. Vanakker, 2023, Frontiers in immunology.

Stereocontrolled access to thioisosteres of nucleoside di- and triphosphates.

Martin D. Eastgate, J. Kowalska, J. Jemielity, 2023, Nature chemistry.