Yoshikazu Sasaki

发表

Synthesis of (Z)-alkene-containing cis-proline dipeptide mimetics using samarium(II) diiodide (SmI2)-mediated reductive alkylation reaction

A. Otaka, N. Fujii, Akira Shigenaga, 2007 .

SmI2-Mediated Reduction of γ,γ-Difluoro-α,β-enoates with Application to the Synthesis of Functionalized (Z)-Fluoroalkene-Type Dipeptide Isosteres

T. Kinoshita, A. Otaka, H. Tamamura, 2004 .

Application of samarium diiodide (SmI2)-induced reduction of γ-acetoxy-α,β-enoates with α-specific kinetic electrophilic trapping for the synthesis of amino acid derivatives

A. Otaka, H. Tamamura, N. Fujii, 2003 .

Asymmetric total synthesis of vindorosine, vindoline, and key vinblastine analogues.

D. Boger, Daisuke Kato, Dale L. Boger, 2010, Journal of the American Chemical Society.

Development of copper-mediated allylation of γ-activated-α,β-unsaturated lactam toward peptide mimetic synthesis

A. Otaka, N. Fujii, Akira Shigenaga, 2007 .

Asymmetric total synthesis of vindoline.

D. Boger, D. Kato, Yoshikazu Sasaki, 2010, Journal of the American Chemical Society.

Reduction of peptide character of HIV protease inhibitors that exhibit nanomolar potency against multidrug resistant HIV-1 strains.

H. Mitsuya, K. Maeda, A. Otaka, 2003, Journal of medicinal chemistry.

Stereoselective synthesis of 3,6-disubstituted-3,6-dihydropyridin-2-ones as potential diketopiperazine mimetics using organocopper-mediated anti-SN2' reactions and their use in the preparation of low-molecule CXCR4 antagonists.

K. Kitaura, A. Otaka, H. Tamamura, 2006, The Journal of organic chemistry.

Total synthesis and evaluation of vinblastine analogues containing systematic deep-seated modifications in the vindoline subunit ring system: core redesign.

Katharine K. Duncan, D. Boger, Annie Tam, 2013, Journal of medicinal chemistry.

Stereoselective synthesis of (Z)-alkene-containing proline dipeptide mimetics.

A. Otaka, N. Fujii, Akira Shigenaga, 2006, The Journal of organic chemistry.

Comparison of one‐pot and two‐step polymerization of polyimide from BPDA/ODA

T. Ogawa, H. Inoue, Yoshikazu Sasaki, 1996 .

Identification of novel benzimidazole derivatives as highly potent AMPK activators with anti-diabetic profiles.

T. Iwasaki, E. Kojima, Y. Hinata, 2022, Bioorganic & medicinal chemistry letters.

Facile access to (Z)-alkene-containing diketopiperazine mimetics utilizing organocopper-mediated anti-SN2′ reactions

A. Otaka, H. Tamamura, N. Fujii, 2005 .

Asymmetric total synthesis of vindoline.

D. Boger, D. Kato, Yoshikazu Sasaki, 2010, Journal of the American Chemical Society.