E. H. Sessions

发表

Synthesis and physicochemical characterization of novel phenotypic probes targeting the nuclear factor-kappa B signaling pathway

John Calvin Reed, G. Roth, R. G. Correa, 2013, Beilstein journal of organic chemistry.

Identification of Inhibitors of NOD1-Induced Nuclear Factor-κB Activation

John Calvin Reed, Brock T Brown, G. Roth, 2011, ACS medicinal chemistry letters.

Discovery and optimization of indoles and 7-azaindoles as Rho kinase (ROCK) inhibitors (part-I).

P. Lograsso, S. Schürer, J. Pocas, 2011, Bioorganic & medicinal chemistry letters.

Synthesis and biological evaluation of 4-quinazolinones as Rho kinase inhibitors.

P. Lograsso, J. Pocas, Yan Yin, 2011, Bioorganic & medicinal chemistry letters.

The development of benzimidazoles as selective rho kinase inhibitors.

P. Lograsso, J. Pocas, Yan Yin, 2010, Bioorganic & Medicinal Chemistry Letters.

Benzimidazole- and benzoxazole-based inhibitors of Rho kinase.

P. Lograsso, S. Schürer, J. Pocas, 2008, Bioorganic & medicinal chemistry letters.

Optimization of a Urea-containing Series of Nicotinamide Phosphoribosyltransferase (NAMPT) Activators.

M. Jackson, E. Sergienko, S. Gardell, 2021, Bioorganic & medicinal chemistry letters.

Measurement of Pyridine Nucleotides in Biological Samples Using LC-MS/MS.

C. Petucci, S. Gardell, D. Divlianska, 2019, Methods in molecular biology.

Discovery of 1-[2-(1-methyl-1H-pyrazol-5-yl)-[1,2,4]triazolo[1,5-a]pyridin-6-yl]-3-(pyridin-4-ylmethyl)urea as a potent NAMPT (nicotinamide phosphoribosyltransferase) activator with attenuated CYP inhibition.

E. Sergienko, M. Yokoyama, S. Gardell, 2021, Bioorganic & medicinal chemistry letters.

Studies on the synthesis of furanosteroids. I. Viridin models.

P. Jacobi, E. H. Sessions, E. H. Sessions, 2006, Organic letters.

Studies on inducers of nerve growth factor: synthesis of the cyathin core.

I. Ghiviriga, D. Wright, D. Frey, 1999, Organic letters.

Two-step electrochemical annulation for the assembly of polycyclic systems.

I. Ghiviriga, D. Wright, C. R. Whitehead, 2002, Organic letters.

Discovery of Novel Small-Molecule Inducers of Heme Oxygenase-1 That Protect Human iPSC-Derived Cardiomyocytes from Oxidative Stress

Siobhan Malany, Patrick Maloney, Layton H. Smith, 2018, The Journal of Pharmacology and Experimental Therapeutics.

Molecular mechanism of a covalent allosteric inhibitor of SUMO E1 activating enzyme

S. Olsen, C. Davies, D. Divlianska, 2018, Nature Communications.

Molecular mechanism of a covalent allosteric inhibitor of SUMO E1 activating enzyme

S. Olsen, C. Davies, D. Divlianska, 2018, Nature Communications.

Constructing the Heterocyclic Core of Viridin and Wortmannin

P. Jacobi, E. O. Onyango, E. H. Sessions, 2013 .

Furanosteroid studies. Stereoselective synthesis of the A,B,E-ring core of wortmannin.

P. Jacobi, E. H. Sessions, R. T. O'Connor, 2007, Organic letters.

Structure-Guided Strategy for the Development of Potent Bivalent ERK Inhibitors.

G. Roth, B. C. Lechtenberg, E. Pasquale, 2017, ACS medicinal chemistry letters.

Crystal structure of SUMO E1 in complex with an allosteric inhibitor

S. Olsen, C. Davies, D. Divlianska, 2018 .

Molecular mechanism of a covalent allosteric inhibitor of SUMO E1 activating enzyme

S. Olsen, C. Davies, D. Divlianska, 2018, Nature Communications.

Identification and characterization of small molecule inhibitors of the ubiquitin ligases Siah1/2 in melanoma and prostate cancer cells.

R. Liddington, M. Jackson, M. Gleave, 2019, Cancer letters.

Discovery of Novel Small-Molecule Inducers of Heme Oxygenase-1 That Protect Human iPSC-Derived Cardiomyocytes from Oxidative Stress

D. Divlianska, Ada Koo, Kevin H. Nguyen, 2018, The Journal of Pharmacology and Experimental Therapeutics.

Boosting NAD+ with a small molecule that activates NAMPT

E. Sergienko, C. Petucci, S. Gardell, 2019, Nature Communications.

Structure-Guided Strategy for the Development of Potent Bivalent ERK Inhibitors.

B. C. Lechtenberg, R. Stalder, Y. Wallez, 2017, ACS medicinal chemistry letters.