T. J. Schrøder

Novel aza-analogous ergoline derived scaffolds as potent serotonin 5-HT₆ and dopamine D₂ receptor ligands.

J. Kehler, C. Christoffersen, N. Krogsgaard‐Larsen, 2014, Journal of medicinal chemistry.

The identification of AF38469: an orally bioavailable inhibitor of the VPS10P family sorting receptor Sortilin.

M. Langgård, C. Bundgaard, J. Stavenhagen, 2014, Bioorganic & medicinal chemistry letters.

Identification of the first small-molecule ligand of the neuronal receptor sortilin and structure determination of the receptor–ligand complex

M. Langgård, S. Thirup, M. Garcia-Alai, 2014, Acta crystallographica. Section D, Biological crystallography.

Discovery of phosphoric acid mono-{2-[(E/Z)-4-(3,3-dimethyl-butyrylamino)-3,5-difluoro-benzoylimino]-thiazol-3-ylmethyl} ester (Lu AA47070): a phosphonooxymethylene prodrug of a potent and selective hA(2A) receptor antagonist.

M. Langgård, C. Bundgaard, B. Bang-Andersen, 2011, Journal of medicinal chemistry.

Synthesis and SAR studies of analogues of 4-(3,3-dimethyl-butyrylamino)-3,5-difluoro-N-thiazol-2-yl-benzamide (Lu AA41063) as adenosine A2A receptor ligands with improved aqueous solubility.

M. Langgård, B. Bang-Andersen, M. Kreilgaard, 2015, Bioorganic & medicinal chemistry letters.

Hit-to-lead optimization of a series of carboxamides of ethyl 2-amino-4-phenylthiazole-5-carboxylates as novel adenosine A2A receptor antagonists.

B. Bang-Andersen, L. Torup, L. Brennum, 2010, Bioorganic & medicinal chemistry letters.

Novel aza-analogous ergoline derived scaffolds as potent serotonin 5-HT₆ and dopamine D₂ receptor ligands.

J. Kehler, C. Christoffersen, N. Krogsgaard‐Larsen, 2014, Journal of medicinal chemistry.