P. Greenspan

发表

Identification of dipeptidyl nitriles as potent and selective inhibitors of cathepsin B through structure-based drug design.

R. Bohacek, H. Zhou, K. Clark, 2001, Journal of medicinal chemistry.

Identification of Novel Carbocyclic Pyrimidine Cyclic Dinucleotide STING Agonists for Antitumor Immunotherapy Using Systemic Intravenous Route.

Adnan O. Abu-Yousif, M. Mizutani, Courtney A. Cullis, 2021, Journal of medicinal chemistry.

Triphenylsilanol as a water surrogate for regioselective Pd catalyzed allylations

B. Trost, P. Greenspan, Nobuhiko Ito, 1993 .

Discovery and optimization of pyrazoline compounds as B-Raf inhibitors.

S. Langston, K. Garcia, C. Blackburn, 2010, Bioorganic & medicinal chemistry letters.

Triphenylsilanol as a Water Surrogate for Regioselective Pd‐Catalyzed Allylations.

B. Trost, P. Greenspan, Nobuhiko Ito, 1993 .

Diastereoselective diels-alder reactions between substituted 1,3-butadienes and n-α-methylbenzylmaleimide

A. McPhail, S. Baldwin, P. Greenspan, 1991 .

A small-molecule inhibitor of the ubiquitin activating enzyme for cancer treatment

S. Tirrell, J. Newcomb, T. Soucy, 2018, Nature Medicine.

Discovery of TAK-981, a First-in-Class Inhibitor of SUMO-Activating Enzyme for the Treatment of Cancer.

Xingyue He, M. Mizutani, T. Soucy, 2021, Journal of medicinal chemistry.

Optimization of tetrahydronaphthalene inhibitors of Raf with selectivity over hERG.

S. Adhikari, H. Mizutani, Mansoureh Rezaei, 2016, Bioorganic & medicinal chemistry letters.

A Total Synthesis of ( + )‐2′S, 3′R‐Zoapatanol

B. Trost, N. Greeves, H. Geissler, 1994 .

Total Synthesis of (+)-(2′S,3′R)-Zoapatanol.

J. H. Kim, B. Trost, N. Greeves, 1995 .

N-arylaminonitriles as bioavailable peptidomimetic inhibitors of cathepsin B.

R. Tommasi, D. Farley, S. Cowen, 2003, Bioorganic & medicinal chemistry letters.

Carboxy-substituted cinnamides: a novel series of potent, orally active LTB4 receptor antagonists.

R. Fujimoto, R. Pelletier, K. Lipson, 1999, Journal of Medicinal Chemistry.

Design and optimization of potent and orally bioavailable tetrahydronaphthalene Raf inhibitors.

Yuan Tian, Hongbo Zeng, Mansoureh Rezaei, 2011, Journal of medicinal chemistry.

An Unusual Oxidative Cyclization. A Synthesis and Absolute Stereochemical Assignment of (-)-Rocaglamide.

B. Trost, B. Yang, G. SaulnierMark, 1991 .

LTB4-induced transient neutropenia in the rat: a model for evaluating efficacy and bioavailability of LTB4 receptor antagonists.

G. Dipasquale, G. Pastor, T. Pellas, 1993, Journal of pharmacological and toxicological methods.