G. Cervi

Discovery of 2-(cyclohexylmethylamino)pyrimidines as a new class of reversible valosine containing protein inhibitors.

A. Isacchi, E. Felder, R. D'Alessio, 2014, Journal of medicinal chemistry.

Bicyclic carbohydrate-derived scaffolds for combinatorial libraries.

F. Nicotra, F. Peri, C. Gennari, 2006, Bioorganic & medicinal chemistry.

Use of multicomponent, domino, and other one-pot syntheses on solid phase: powerful tools for the generation of libraries of diverse and complex compounds.

M. Pulici, K. Martina, F. Quartieri, 2003, Combinatorial chemistry & high throughput screening.

Identification of N,1,4,4-tetramethyl-8-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4,5-dihydro-1H-pyrazolo[4,3-h]quinazoline-3-carboxamide (PHA-848125), a potent, orally available cyclin dependent kinase inhibitor.

A. Isacchi, E. Casale, C. Mercurio, 2009, Journal of medicinal chemistry.

Thieno[3,2-c]pyrazoles: a novel class of Aurora inhibitors with favorable antitumor activity.

V. Croci, D. Volpi, F. Roletto, 2010, Bioorganic & medicinal chemistry.

Covalent and allosteric inhibitors of the ATPase VCP/p97 induce cancer cell death.

A. Isacchi, E. Casale, Daniel J. Anderson, 2013, Nature chemical biology.

Discovery and optimization of pyrrolo[1,2-a]pyrazinones leads to novel and selective inhibitors of PIM kinases.

E. Casale, E. Felder, A. Galvani, 2013, Bioorganic & medicinal chemistry.