Christian Ragot

New Potent DOT1L Inhibitors for in Vivo Evaluation in Mouse.

R. Tiedt, D. Guthy, C. Scheufler, 2019, ACS medicinal chemistry letters.

Discovery of Potent, Selective, and Structurally Novel Dot1L Inhibitors by a Fragment Linking Approach.

Philipp Holzer, R. Tiedt, G. Caravatti, 2017, ACS medicinal chemistry letters.

Optimization of a Fragment-Based Screening Hit toward Potent DOT1L Inhibitors Interacting in an Induced Binding Pocket.

R. Tiedt, C. Fernández, C. Scheufler, 2016, ACS medicinal chemistry letters.