H. Miyazoe

发表

Discovery of novel arylpyrazole series as potent and selective opioid receptor-like 1 (ORL1) antagonists.

S. Ozaki, Y. Ishii, Yasushi Nagatomi, 2009, Bioorganic & medicinal chemistry letters.

Convergent synthesis of silylated allylic alcohols by a stereoselective domino, sequential radical-coupling reaction.

J. Yoshida, S. Yamago, H. Miyazoe, 2002, Angewandte Chemie.

Reversible generation of glycosyl radicals from telluroglycosides under photochemical and thermal conditions

J. Yoshida, S. Yamago, H. Miyazoe, 1999 .

Design, synthesis, and structure-activity relationship study of a novel class of ORL1 receptor antagonists based on N-biarylmethyl spiropiperidine.

S. Ozaki, H. Ohta, Masanori Asai, 2008, Bioorganic & medicinal chemistry letters.

Synthetic and theoretical studies on group-transfer imidoylation of organotellurium compounds. remarkable reactivity of isonitriles in comparison with carbon monoxide in radical-mediated reactions.

S. Yamago, J. Yoshida, M. Hashidume, 2001, Journal of the American Chemical Society.

Novel Group‐Transfer Three‐Component Coupling of Silyltellurides, Carbonyl Compounds, and Isocyanides

J. Yoshida, S. Yamago, H. Miyazoe, 2000 .

New synthesis of α-acyl imines by radical-mediated group-transfer imidoylation of acyl tellurides with isonitriles

J. Yoshida, S. Yamago, T. Sawazaki, 2000 .

Radical-mediated imidoylation of telluroglycosides. Insertion of isonitriles into the glycosidic carbontellurium bond

J. Yoshida, S. Yamago, H. Miyazoe, 1999 .

Synthesis of vinylic C-glycosides from telluroglycosides. Addition of photochemically and thermally generated glycosyl radicals to alkynes

J. Yoshida, S. Yamago, H. Miyazoe, 1999 .

A diversity-oriented synthesis of alpha-amino acid derivatives by a silyltelluride-mediated radical coupling reaction of imines and isonitriles.

J. Yoshida, S. Yamago, H. Miyazoe, 2003, Angewandte Chemie.

A novel class of cycloalkano[b]pyridines as potent and orally active opioid receptor-like 1 antagonists with minimal binding affinity to the hERG K+ channel.

Hisashi Ohta, Hiroshi Kawamoto, Satoshi Ozaki, 2008, Journal of medicinal chemistry.

Synthetic and Theoretical Studies on Group‐Transfer Imidoylation of Organotellurium Compounds. Remarkable Reactivity of Isonitriles in Comparison with Carbon Monoxide in Radical‐Mediated Reactions.

J. Yoshida, S. Yamago, M. Hashidume, 2001 .

Radical-Mediated Imidoylation of Telluroglycosides. Insertion of Isonitriles into the Glycosidic Carbon—Tellurium Bond.

J. Yoshida, S. Yamago, H. Miyazoe, 1999 .

Discovery of novel diarylketoxime derivatives as selective and orally active melanin-concentrating hormone 1 receptor antagonists.

Kouta Masutani, M. Kameda, H. Matsushita, 2009, Bioorganic & medicinal chemistry letters.

2-Cyclohexylcarbonylbenzimidazoles as potent, orally available and brain-penetrable opioid receptor-like 1 (ORL1) antagonists.

Hisashi Ohta, Hiroshi Kawamoto, Satoshi Ozaki, 2009, Bioorganic & medicinal chemistry letters.

Optimization of a series of 2,4-diaminopyridines as neuropeptide Y Y1 receptor antagonists with reduced hERG activity.

Tomoki Suzuki, M. Kameda, M. Ando, 2009, Bioorganic & medicinal chemistry letters.

2-Cyclohexylcarbonylbenzimidazoles as potent, orally available and brain-penetrable opioid receptor-like 1 (ORL1) antagonists.

S. Ozaki, Y. Ishii, S. Ito, 2009, Bioorganic & medicinal chemistry letters.

Design, synthesis and evaluation of a novel cyclohexanamine class of neuropeptide Y Y1 receptor antagonists.

Tomoki Suzuki, M. Ando, Kensuke Kobayashi, 2009, Bioorganic & medicinal chemistry letters.