Junya Qu

发表

Discovery of Isoxazole Amides as Potent and Selective SMYD3 Inhibitors.

J. Luengo, A. P. Graves, M. Pappalardi, 2019, ACS medicinal chemistry letters.

Rational Design, Synthesis, and SAR of a Novel Thiazolopyrimidinone Series of Selective PI3K-beta Inhibitors.

J. F. Mack, J. Luengo, Ramona N Plant, 2012, ACS medicinal chemistry letters.

[3a,4]-Dihydropyrazolo[1,5a]pyrimidines: Novel, Potent, and Selective Phosphatidylinositol-3-kinase β Inhibitors.

J. Luengo, Ramona N Plant, K. Erhard, 2013, ACS medicinal chemistry letters.

2-Amino-3,4-dihydroquinazolines as inhibitors of BACE-1 (beta-site APP cleaving enzyme): Use of structure based design to convert a micromolar hit into a nanomolar lead.

Junya Qu, Allen B Reitz, Brett A Tounge, 2007, Journal of medicinal chemistry.

Facile synthesis of 6-aryl 5-N-substituted pyridazinones: microwave-assisted Suzuki-Miyaura cross coupling of 6-chloropyridazinones.

G. Burton, R. Rivero, P. Cao, 2008, The Journal of organic chemistry.

Imino Ene Reactions of Enantiopure N-Sulfinylimino Esters: Asymmetric Synthesis of 1-Oxo-1 λ4-isothiazolidine-3-carboxylates

R. Joseph, F. A. Davis, D. D. Titus, 2002 .

Discovery and characterization of a cell-permeable, small-molecule c-Abl kinase activator that binds to the myristoyl binding site.

Yoshiaki Washio, Junya Qu, Thau Ho, 2011, Chemistry & biology.

Structure-guided optimization of small molecule c-Abl activators

Ping Cao, Jingsong Yang, Hong Zhang, 2014, Journal of Computer-Aided Molecular Design.

Discovery of a Novel 2,6-Disubstituted Glucosamine Series of Potent and Selective Hexokinase 2 Inhibitors.

Yong Jiang, Jacques Briand, Junya Qu, 2016, ACS medicinal chemistry letters.

Discovery and characterization of a cell-permeable, small-molecule c-Abl kinase activator that binds to the myristoyl binding site.

M. Head, S. Moores, G. Hofmann, 2011, Chemistry & biology.