A. Lukin

发表

Novel FFA1 (GPR40) agonists containing spirocyclic periphery: polar azine periphery as a driver of potency

S. Zozulya, M. Krasavin, I. Zahanich, 2016, Journal of enzyme inhibition and medicinal chemistry.

Novel agonists of free fatty acid receptor 1 (GPR40) based on 3-(1,3,4-thiadiazol-2-yl)propanoic acid scaffold

S. Zozulya, M. Krasavin, I. Zahanich, 2016, Journal of enzyme inhibition and medicinal chemistry.

Discovery and In Vivo Efficacy of Trace Amine-Associated Receptor 1 (TAAR1) Agonist 4-(2-Aminoethyl)-N-(3,5-dimethylphenyl)piperidine-1-carboxamide Hydrochloride (AP163) for the Treatment of Psychotic Disorders

R. Gainetdinov, M. Krasavin, Anatoly A. Peshkov, 2022, International journal of molecular sciences.

Spirocyclic amino alcohol building blocks prepared via a Prins-type cyclization in aqueous sulfuric acid

M. Krasavin, A. Lukin, N. Zhurilo, 2016 .

Discovery of polar spirocyclic orally bioavailable urea inhibitors of soluble epoxide hydrolase.

J. Leppänen, E. Proschak, S. Auriola, 2018, Bioorganic chemistry.

Zn-catalyzed hydrohydrazination of propargylamides with BocNHNH2: a novel entry into the 1,2,4-triazine core

M. Krasavin, D. Tovpeko, A. Lukin, 2016 .

Zn-Catalyzed Hydrohydrazination of Propargylamides with BocNHNH2: A Novel Entry into the 1,2,4-Triazine Core.

M. Krasavin, D. Tovpeko, A. Lukin, 2016 .

Polar aromatic periphery increases agonist potency of spirocyclic free fatty acid receptor (GPR40) agonists inspired by LY2881835.

I. Tikhonova, S. Zozulya, A. Golovanov, 2017, European journal of medicinal chemistry.

Discovery of Trace Amine-Associated Receptor 1 (TAAR1) Agonist 2-(5-(4′-Chloro-[1,1′-biphenyl]-4-yl)-4H-1,2,4-triazol-3-yl)ethan-1-amine (LK00764) for the Treatment of Psychotic Disorders

R. Gainetdinov, M. Krasavin, M. Gureev, 2022, Biomolecules.

Exploration of the nitrogen heterocyclic periphery around the core of the advanced FFA1 agonist fasiglifam (TAK‐875)

S. Zozulya, O. Onopchenko, M. Krasavin, 2020, Archiv der Pharmazie.

Free fatty acid receptor 1 (GPR40) agonists containing spirocyclic periphery inspired by LY2881835.

I. Tikhonova, M. Lehtonen, J. Rautio, 2016, Bioorganic & medicinal chemistry.

Novel free fatty acid receptor 1 (GPR40) agonists based on 1,3,4-thiadiazole-2-carboxamide scaffold.

I. Tikhonova, S. Zozulya, M. Krasavin, 2016, Bioorganic & medicinal chemistry.

Identification of a novel trace amine-associated receptor 1 agonist with in vivo activity

R. Gainetdinov, M. Krasavin, M. Dorofeikova, 2018, European Neuropsychopharmacology.

Synthesis of radicals underlain by 1,3-bis(4,5-diphenylimidazol-2-yl)benzene

A. V. Dolganov, B. Tanaseichuk, M. K. Pryanichnikova, 2011 .

Synthesis of 1-oxa-9-azaspiro[5.5]undecane-9-sulfonamides bearing a diverse molecular periphery and a rare zinc-binding group for carbonic anhydrase interrogation

S. Kalinin, M. Krasavin, A. Lukin, 2023, Mendeleev Communications.

Discovery of Trace Amine-Associated Receptor 1 (TAAR1) Agonist 2-(5-(4'-Chloro-[1,1'-biphenyl]-4-yl)-4H-1,2,4-triazol-3-yl)ethan-1-amine (LK00764) for the Treatment of Psychotic Disorders

R. Gainetdinov, M. Krasavin, M. Gureev, 2022 .

Spirocyclic azetidines for drug discovery: Novel Boc-protected 7'H-spiro[azetidine-3,5'-furo[3,4-d ]pyrimidines]

M. Krasavin, A. Lukin, Lyubov V. Vinogradova, 2023, Mendeleev Communications.

5-Nitrofuran-2-yl Thiohydrazones as Double Antibacterial Agents Synthesis and In Vitro Evaluation

M. Chudinov, A. Lukin, T. Vedekhina, 2020 .

Polar aromatic periphery increases agonist potency of spirocyclic free fatty acid receptor (GPR40) agonists inspired by LY2881835.

I. Tikhonova, S. Zozulya, A. Golovanov, 2017, European journal of medicinal chemistry.