Sang-Uk Kang

发表

Synthesis of tripeptides as potent Yersinia protein tyrosine phosphatase inhibitors.

K. No, Ky-Youb Nam, Zhon-Yin Zhang, 2005, Bioorganic & medicinal chemistry letters.

A one-step synthesis of Nα-Fmoc-4-O-[O′,O″-di-tert-butyl-2-(2-fluoromalonyl)]-l-tyrosine from commercially available starting material

T. Burke, Sang-Uk Kang, 2004 .

1,2,4-Triazole fused heterocycles by electrocyclic reaction of N-aziridinylimino carbodiimides obtained from N-aziridinylimino ureas

K. Lee, Sang-Uk Kang, 1995 .

N-[4-(methylsulfonylamino)benzyl]thiourea analogues as vanilloid receptor antagonists: analysis of structure-activity relationships for the "C-Region".

Jeewoo Lee, P. Blumberg, L. Pearce, 2004, Bioorganic & medicinal chemistry.

N-(3-acyloxy-2-benzylpropyl)-N'-[4-(methylsulfonylamino)benzyl]thiourea analogues: novel potent and high affinity antagonists and partial antagonists of the vanilloid receptor.

Ji-Min Kim, Attila Toth, Jiyoun Lee, 2003, Journal of medicinal chemistry.

Novel potent antagonists of transient receptor potential channel, vanilloid subfamily member 1: structure-activity relationship of 1,3-diarylalkyl thioureas possessing new vanilloid equivalents.

Jin Kwan Kim, S. Shin, Kwang-Ok Lee, 2005, Journal of medicinal chemistry.

Analysis of structure-activity relationships for the 'A-region' of N-(4-t-butylbenzyl)-N'-[4-(methylsulfonylamino)benzyl]thiourea analogues as TRPV1 antagonists.

Vladimir A. Pavlyukovets, S. Y. Kim, Jeewoo Lee, 2005, Bioorganic & medicinal chemistry letters.

Analysis of structure-activity relationships for the 'B-region' of N-(4-t-butylbenzyl)-N'-[4-(methylsulfonylamino)benzyl]-thiourea analogues as TRPV1 antagonists.

Vladimir A. Pavlyukovets, Jiyoun Lee, S. Y. Kim, 2005, Bioorganic & medicinal chemistry letters.

GPR119 agonists: a promising approach for T2DM treatment? A SWOT analysis of GPR119.

Sang-Uk Kang, Sang-Uk Kang, 2013, Drug discovery today.

Analysis of structure-activity relationships for the 'B-region' of N-(3-acyloxy-2-benzylpropyl)-N(')-[4-(methylsulfonylamino)benzyl]thiourea analogues as vanilloid receptor antagonists: discovery of an N-hydroxythiourea analogue with potent analgesic activity.

Jeewoo Lee, P. Blumberg, Kang-Pil Kim, 2004, Bioorganic & medicinal chemistry letters.

Synthesis of α,α-disubstituted 4-phosphonophenylalanine analogues as conformationally-constrained phosphotyrosyl mimetics

J. Deschamps, Dajun Yang, Manchao Zhang, 2004 .

N-Alkoxysulfamide, N-hydroxysulfamide, and sulfamate analogues of methionyl and isoleucyl adenylates as inhibitors of methionyl-tRNA and isoleucyl-tRNA synthetases.

S. Y. Kim, Taehee Kang, Jeewoo Lee, 2003, Bioorganic & medicinal chemistry letters.

High affinity antagonists of the vanilloid receptor.

Jiyoun Lee, P. Blumberg, Y. Suh, 2002, Molecular pharmacology.

High-affinity partial agonists of the vanilloid receptor.

P. Blumberg, A. Tóth, Richard Tran, 2003, Molecular pharmacology.

Structure-activity relationships of simplified resiniferatoxin analogues with potent VR1 agonism elucidates an active conformation of RTX for VR1 binding.

S. Y. Kim, Jeewoo Lee, P. Blumberg, 2004, Bioorganic & medicinal chemistry.

N-4-Substituted-benzyl-N'-tert-butylbenzyl thioureas as vanilloid receptor ligands: investigation on the role of methanesulfonamido group in antagonistic activity.

Y. Suh, H. Kim, Hyeung‐geun Park, 2004, Bioorganic & medicinal chemistry letters.

Different vanilloid agonists cause different patterns of calcium response in CHO cells heterologously expressing rat TRPV1.

P. Blumberg, Yun Wang, L. Pearce, 2005, Life sciences.

Alpha-substituted N-(4-tert-butylbenzyl)-N'-[4-(methylsulfonylamino)benzyl]thiourea analogues as potent and stereospecific TRPV1 antagonists.

Vladimir A. Pavlyukovets, Sun Choi, S. Y. Kim, 2007, Bioorganic & medicinal chemistry.

Examination of acylated 4-aminopiperidine-4-carboxylic acid residues in the phosphotyrosyl+1 position of Grb2 SH2 domain-binding tripeptides.

R. Fisher, T. Burke, W. J. Choi, 2007, Journal of Medicinal Chemistry.

Stereospecific high-affinity TRPV1 antagonists: chiral N-(2-benzyl-3-pivaloyloxypropyl) 2-[4-(methylsulfonylamino)phenyl]propionamide analogues.

Dong Wook Kang, Attila Toth, HyungChul Ryu, 2008, Journal of medicinal chemistry.

Design and synthesis of conformationally constrained Grb2 SH2 domain binding peptides employing alpha-methylphenylalanyl based phosphotyrosyl mimetics.

Marc C Nicklaus, Shinya Oishi, Robert J Fisher, 2005, Journal of medicinal chemistry.