B. G. K. Perera

发表

Chemical Proteomic Tools for Studying Protein Kinase Active Sites

B. G. K. Perera, 2012 .

Allosteric Inhibition of the IRE1α RNase Preserves Cell Viability and Function during Endoplasmic Reticulum Stress

Dustin J Maly, E. Snapp, R. Ghosh, 2014, Cell.

Conformation-selective inhibitors reveal differences in the activation and phosphate-binding loops of the tyrosine kinases Abl and Src.

Dustin J Maly, M. Seeliger, S. Hari, 2013, ACS chemical biology.

Multiple determinants for selective inhibition of apicomplexan calcium-dependent protein kinase CDPK1.

Steven M. Johnson, C. Verlinde, W. Hol, 2012, Journal of medicinal chemistry.

Affinity-based probes based on type II kinase inhibitors.

Dustin J Maly, J. Villén, E. Merritt, 2012, Journal of the American Chemical Society.

Allosteric Inhibition of the IRE1a RNase Preserves Cell Viability and Function during Endoplasmic Reticulum Stress

E. Snapp, R. Ghosh, F. R. Papa, 2015 .

Allosteric Inhibition of the IRE 1 a RNase Preserves Cell Viability and Function during Endoplasmic Reticulum Stress

Dustin J Maly, E. Snapp, R. Ghosh, 2014 .

Bivalent inhibitors of the tyrosine kinases ABL and SRC: determinants of potency and selectivity.

Dustin J Maly, Z. Hill, B. G. K. Perera, 2011, Molecular bioSystems.

Design, synthesis and characterization of "clickable" 4-anilinoquinazoline kinase inhibitors.

Dustin J Maly, B. G. K. Perera, 2008, Molecular bioSystems.

Targeting diverse signaling interaction sites allows the rapid generation of bivalent kinase inhibitors.

Simeon S. Andrews, Dustin J Maly, Z. Hill, 2012, ACS chemical biology.

ATP-Competitive Partial Antagonists of IRE1α’s RNase Segregate Outputs of the UPR

R. Ghosh, F. R. Papa, J. Zikherman, 2021, Nature Chemical Biology.

A hexylchloride-based catch-and-release system for chemical proteomic applications.

Dustin J Maly, Jennifer L Brigham, B. G. K. Perera, 2013, ACS chemical biology.

Divergent allosteric control of the IRE1α endoribonuclease using kinase inhibitors

Dustin J Maly, F. R. Papa, M. Seeliger, 2012, Nature chemical biology.

Development of Toxoplasma gondii calcium-dependent protein kinase 1 (TgCDPK1) inhibitors with potent anti-toxoplasma activity.

Steven M. Johnson, Dustin J Maly, M. Parsons, 2012, Journal of medicinal chemistry.

Biolayer Interferometry Assay for Cyclin-Dependent Kinase-Cyclin Association Reveals Diverse Effects of Cdk2 Inhibitors on Cyclin Binding Kinetics.

Dustin J Maly, G. Kiss, A. Bridges, 2023, ACS chemical biology.

Discovery of Potent and Selective Inhibitors of CDPK1 from C. parvum and T. gondii

Dustin J Maly, W. V. Voorhis, C. Verlinde, 2010 .

A chemical genetic method for generating bivalent inhibitors of protein kinases.

Dustin J Maly, Z. Hill, B. G. K. Perera, 2009, Journal of the American Chemical Society.

Label Transfer Reagents to Probe p38 MAPK Binding Partners

Simeon S. Andrews, Dustin J Maly, Z. Hill, 2013, Chembiochem : a European journal of chemical biology.

Discovery of Potent and Selective Inhibitors of Calcium-Dependent Protein Kinase 1 (CDPK1) from C. parvum and T. gondii.

Dustin J Maly, C. Verlinde, E. Merritt, 2010, ACS medicinal chemistry letters.

A Compound that Inhibits Glycolysis in Prostate Cancer Controls Growth of Advanced Prostate Cancer

Dustin J Maly, Shihua Sun, S. Plymate, 2023, bioRxiv.

A Compound that Inhibits Glycolysis in Prostate Cancer Controls Growth of Advanced Prostate Cancer.

Dustin J Maly, S. Plymate, Lucas B. Sullivan, 2024, Molecular cancer therapeutics.

A Compound that Inhibits Glycolysis in Prostate Cancer Controls Growth of Advanced Prostate Cancer

Dustin J Maly, S. Plymate, Lucas B. Sullivan, 2023, bioRxiv.