M. Nagamochi

发表

Design, Synthesis, and Biological Evaluation of Novel 7-[(3 aS,7 aS)-3 a-Aminohexahydropyrano[3,4- c]pyrrol-2(3 H)-yl]-8-methoxyquinolines with Potent Antibacterial Activity against Respiratory Pathogens.

Hisashi Takahashi, T. Kitamura, S. Komoriya, 2018, Journal of medicinal chemistry.

Stereoselective synthesis and biological evaluation of 3,4-diaminocyclohexanecarboxylic acid derivatives as factor Xa inhibitors.

Tsutomu Nagata, H. Kanno, T. Yoshino, 2008, Bioorganic & Medicinal Chemistry Letters.

Discovery of N-[(1R,2S,5S)-2-{[(5-chloroindol-2-yl)carbonyl]amino}-5-(dimethylcarbamoyl)cyclohexyl]-5-methyl-4,5,6,7-tetrahydrothiazolo[5,4-c]pyridine-2-carboxamide hydrochloride: a novel, potent and orally active direct inhibitor of factor Xa.

N. Haginoya, Makoto Suzuki, Tsutomu Nagata, 2009, Bioorganic & medicinal chemistry.

A general and practical method of alkynyl indole and benzofuran synthesis via tandem Cu- and Pd-catalyzed cross-couplings.

M. Lautens, Yuan-Qing Fang, M. Nagamochi, 2007, Organic letters.

A concise and enantioselective approach to cyclobutanones by tandem asymmetric epoxidation and enantiospecific ring expansion of cyclopropylidene alcohols. An enantiocontrolled synthesis of (+)-and (-)-α-cuparenones

H. Nemoto, K. Fukumoto, M. Nagamochi, 1992 .

A remarkable substituent effect on the enantioselectivity of tandem asymmetric epoxidation and enantiospecific ring expansion of cyclopropylidene alcohols: a new enantiocontrolled synthesis of (-)-debromoaplysin and (-)-aplysin

H. Nemoto, K. Fukumoto, M. Nagamochi, 1994 .

Chiral cyclobutanones as versatile synthons: the first enantioselective total synthesis of (+)-laurene

H. Nemoto, K. Fukumoto, M. Nagamochi, 1993 .

An Enantiocontrolled Formal Total Synthesis of (+)-Ipomeamarone, (-)-Ngaione, and Their Epimers

T. Tanabe, H. Nemoto, K. Fukumoto, 1993 .

A general and practical method of alkynyl indole and benzofuran synthesis via tandem Cu- and Pd-catalyzed cross-couplings.

M. Lautens, Yuan-Qing Fang, M. Nagamochi, 2007, Organic letters.

The first enantioselective total synthesis of (+)-laurene

H. Nemoto, K. Fukumoto, M. Nagamochi, 1992 .

Design, synthesis, and biological evaluations of novel 7-[7-amino-7-methyl-5-azaspiro[2.4]heptan-5-yl]-8-methoxyquinolines with potent antibacterial activity against respiratory pathogens.

Hisashi Takahashi, Y. Sugimoto, J. Kuroyanagi, 2013, Journal of medicinal chemistry.

A novel and efficient route to chiral A-ring aromatic trichothecanes—The first enantiocontrolled total synthesis of (-)-debromofiliformin and (-)-filiformin

H. Hakamata, H. Nemoto, K. Fukumoto, 1995 .

Facile Methods for Preparation of Thiazolopyridine and Tetrahydro-thiazolopyridine Derivatives

N. Haginoya, Tsutomu Nagata, H. Kanno, 2004 .

Facile Methods for Preparation of Thiazolopyridine and Tetrahydrothiazolopyridine Derivatives.

N. Haginoya, Tsutomu Nagata, H. Kanno, 2004 .

Lead optimization of pyrido[2,3-d][1]benzazepin-6-one derivatives leading to the discovery of a potent, selective, and orally available human parathyroid hormone receptor 1 (hPTHR1) antagonist (DS69910557).

Masanori Izumi, Y. Arai, Y. Kiyotsuka, 2022, Bioorganic & medicinal chemistry.

Discovery of novel, potent, and orally bioavailable pyrido[2,3-d][1]benzazepin-6-one antagonists for parathyroid hormone receptor 1.

T. Nishi, Masanori Izumi, Y. Arai, 2020, Bioorganic & medicinal chemistry.