Toshikazu Yokoyama

An expeditious synthesis of tamoxifen, a representative SERM (selective estrogen receptor modulator), via the three-component coupling reaction among aromatic aldehyde, cinnamyltrimethylsilane, and beta-chlorophenetole.

M. Ikekita, Y. Nagahara, Akane Sasaki, 2007, Bioorganic & medicinal chemistry.