Thomas Drapier

Enhancing Action of Positive Allosteric Modulators through the Design of Dimeric Compounds.

J. Kastrup, S. Dilly, B. Pirotte, 2018, Journal of medicinal chemistry.

7-Phenoxy-Substituted 3,4-Dihydro-2H-1,2,4-benzothiadiazine 1,1-Dioxides as Positive Allosteric Modulators of α-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid (AMPA) Receptors with Nanomolar Potency.

P. Tullio, C. Ptak, R. Oswald, 2018, Journal of medicinal chemistry.

Crystal Structures of Potent Dimeric Positive Allosteric Modulators at the Ligand-Binding Domain of the GluA2 Receptor.

J. Kastrup, B. Pirotte, S. Laulumaa, 2018, ACS medicinal chemistry letters.