Lars Jørgensen

发表

Selective mGAT2 (BGT-1) GABA uptake inhibitors: design, synthesis, and pharmacological characterization.

Arne Schousboe, A. Schousboe, P. Krogsgaard‐Larsen, 2013, Journal of medicinal chemistry.

Subunit-Specific Agonist Activity at NR2A-, NR2B-, NR2C-, and NR2D-Containing N-Methyl-d-aspartate Glutamate Receptors

Matthew T. Geballe, J. Snyder, S. Traynelis, 2007, Molecular Pharmacology.

Subunit-Specific Agonist Activity at NR 2 A-, NR 2 B-, NR 2 C-, and NR 2 D-Containing N-Methyl-D-aspartate Glutamate Receptors

Matthew T. Geballe, J. Snyder, S. Traynelis, 2007 .

Discovery of a subtype selective inhibitor of the human betaine/GABA transporter 1 (BGT-1) with a non-competitive pharmacological profile.

A. Schousboe, R. Clausen, H. Bräuner‐Osborne, 2013, Biochemical Pharmacology.

Structural Determinants of Agonist Efficacy at the Glutamate Binding Site of N-Methyl-d-Aspartate Receptors

S. Traynelis, Katie M Vance, Kevin K Ogden, 2013, Molecular Pharmacology.

Structure-Activity Relationship, Pharmacological Characterization, and Molecular Modeling of Noncompetitive Inhibitors of the Betaine/γ-Aminobutyric Acid Transporter 1 (BGT1).

G. Ecker, A. Schousboe, P. Wellendorph, 2017, Journal of medicinal chemistry.

Analogues of 3-Hydroxyisoxazole-Containing Glutamate Receptor Ligands Based on the 3-Hydroxypyrazole-Moiety: Design, Synthesis and Pharmacological Characterization

A. Kristensen, R. Clausen, D. Pickering, 2014, Neurochemical Research.

Analogues of 3-Hydroxyisoxazole-Containing Glutamate Receptor Ligands Based on the 3-Hydroxypyrazole-Moiety: Design, Synthesis and Pharmacological Characterization

A. Kristensen, R. Clausen, D. Pickering, 2014, Neurochemical Research.

Structure activity relationship of selective GABA uptake inhibitors.

G. Ecker, A. Schousboe, R. Clausen, 2015, Bioorganic & medicinal chemistry.

N-Hydroxypyrazolyl glycine derivatives as selective N-methyl-D-aspartic acid receptor ligands.

J. Greenwood, S. Traynelis, K. Hansen, 2008, Journal of medicinal chemistry.

Enzyme kinetic studies of histone demethylases KDM4C and KDM6A: Towards understanding selectivity of inhibitors targeting oncogenic histone demethylases

L. Olsen, J. Kastrup, M. Gajhede, 2011, FEBS letters.