Hannelore Stockhausen

发表

6,6-Fused heterocyclic ureas as highly potent TRPV1 antagonists.

K. Schiene, Sun Choi, Jeewoo Lee, 2015, Bioorganic & medicinal chemistry letters.

2-(3-fluoro-4-methylsulfonylaminophenyl)propanamides as potent transient receptor potential vanilloid 1 (TRPV1) antagonists: structure-activity relationships of 2-amino derivatives in the N-(6-trifluoromethylpyridin-3-ylmethyl) C-region.

Dong Wook Kang, Sun Choi, Mi-Yeon Kim, 2012, Journal of medicinal chemistry.

Discovery of 1-(1H-Indazol-4-yl)-3-((1-Phenyl-1H-Pyrazol-5-yl)methyl) Ureas as Potent and Thermoneutral TRPV1 Antagonists.

G. Bahrenberg, P. Blumberg, Sun-Ok Kwon, 2020, Bioorganic & medicinal chemistry letters.

Discovery of indane propanamides as potent and selective TRPV1 antagonists.

G. Bahrenberg, P. Blumberg, Y. H. Kim, 2019, Bioorganic & medicinal chemistry letters.

Discovery of 2-(3,5-difluoro-4-methylsulfonaminophenyl)propanamides as potent TRPV1 antagonists.

G. Bahrenberg, P. Blumberg, Changhoon Kim, 2018, Bioorganic & medicinal chemistry letters.

t-Butyl pyridine and phenyl C-region analogues of 2-(3-fluoro-4-methylsulfonylaminophenyl)propanamides as potent TRPV1 antagonists.

Sun Choi, G. Bahrenberg, P. Blumberg, 2017, Bioorganic & medicinal chemistry.

Structure activity relationships of benzyl C-region analogs of 2-(3-fluoro-4-methylsulfonamidophenyl)propanamides as potent TRPV1 antagonists.

M. Cui, Sun Choi, G. Bahrenberg, 2015, Bioorganic & medicinal chemistry.

α-Substituted 2-(3-fluoro-4-methylsulfonamidophenyl)acetamides as potent TRPV1 antagonists.

M. Cui, Sun Choi, G. Bahrenberg, 2015, Bioorganic & medicinal chemistry letters.

Pyridine C-region analogs of 2-(3-fluoro-4-methylsulfonylaminophenyl)propanamides as potent TRPV1 antagonists.

HyungChul Ryu, Suyoung Yoon, K. Schiene, 2015, European journal of medicinal chemistry.

In vitro characterization of the thermoneutral transient receptor potential vanilloid-1 (TRPV1) inhibitor GRTE16523.

G. Bahrenberg, N. Damann, Jihyae Ann, 2020, European journal of pharmacology.

4-Aminophenyl acetamides and propanamides as potent transient receptor potential vanilloid 1 (TRPV1) ligands.

Sun Choi, G. Bahrenberg, P. Blumberg, 2018, Bioorganic & medicinal chemistry.

Pyrazole C-region analogues of 2-(3-fluoro-4-methylsulfonylaminophenyl)propanamides as potent TRPV1 antagonists.

Sun Choi, G. Bahrenberg, P. Blumberg, 2017, Bioorganic & medicinal chemistry letters.

2-Alkyl/alkenyl substituted pyridine C-region analogues of 2-(3-fluoro-4-methylsulfonylaminophenyl)propanamides as highly potent TRPV1 antagonists.

K. Schiene, M. Cui, Sun Choi, 2014, Bioorganic & medicinal chemistry letters.

Reduction of myocardial reperfusion injury by an inhibitor of poly (ADP-ribose) synthetase in the pig.

C. Thiemermann, H. Ruetten, P. Martorana, 1998, European journal of pharmacology.