E. Terefenko

发表

Novel 6-aryl-1,4-dihydrobenzo[d]oxazine-2-thiones as potent, selective, and orally active nonsteroidal progesterone receptor agonists.

R. Winneker, Eugene A. Terefenko, J. Wrobel, 2003, Bioorganic & medicinal chemistry letters.

Synthesis and structure-activity relationship of novel 6-aryl-1,4-dihydrobenzo[d][1,3]oxazine-2-thiones as progesterone receptor modulators leading to the potent and selective nonsteroidal progesterone receptor agonist tanaproget.

R. Winneker, R. Chopra, K. Svenson, 2005, Journal of medicinal chemistry.

Potent nonsteroidal progesterone receptor agonists: synthesis and SAR study of 6-aryl benzoxazines.

R. Winneker, J. Wrobel, Zhiming Zhang, 2002, Bioorganic & medicinal chemistry letters.

The reaction of o-amino aryl carboxylic acids with Grignard reagents. The unusual effect of the N-protecting group on aryl ketone formation

Eugene A. Terefenko, Puwen Zhang, E. Terefenko, 2001 .

Thiourea inhibitors of herpes viruses. Part 1: bis-(aryl)thiourea inhibitors of CMV.

S. Lang, K. Curran, B. Feld, 2003, Bioorganic & medicinal chemistry letters.

Thiourea inhibitors of herpes viruses. Part 2: N-Benzyl-N'-arylthiourea inhibitors of CMV.

S. Lang, K. Curran, B. Feld, 2004, Bioorganic & medicinal chemistry letters.

SAR studies of 6-(arylamino)-4,4-disubstituted-1-methyl-1,4-dihydro-benzo[d][1,3]oxazin-2-ones as progesterone receptor antagonists.

R. Winneker, Eugene A. Terefenko, J. Wrobel, 2007, Bioorganic & Medicinal Chemistry Letters.

6-Aryl-1,4-dihydro-benzo[d][1,3]oxazin- 2-ones: a novel class of potent, selective, and orally active nonsteroidal progesterone receptor antagonists.

R. Winneker, S. Lundeen, Eugene A. Terefenko, 2002, Journal of medicinal chemistry.

SAR studies of 6-aryl-1,3-dihydrobenzimidazol-2-ones as progesterone receptor antagonists.

R. Winneker, J. Wrobel, Zhiming Zhang, 2005, Bioorganic & medicinal chemistry letters.

Structure-property relationships that influence platinum stability in all-silica or highly siliceous zeolites

A. Burton, A. Sattler, Michele Paccagnini, 2023, Microporous and Mesoporous Materials.

Structure-activity relationships of the 1-amino-3-(1H-indol-1-yl)-3-phenylpropan-2-ol series of monoamine reuptake inhibitors.

K. Burroughs, D. Deecher, P. Mahaney, 2009, Bioorganic & medicinal chemistry letters.

Synthesis and activity of novel 1- or 3-(3-amino-1-phenyl propyl)-1,3-dihydro-2H-benzimidazol-2-ones as selective norepinephrine reuptake inhibitors.

E. Koury, D. Deecher, P. Mahaney, 2008, Bioorganic & medicinal chemistry letters.

5-(3-Cyclopentyl-2-thioxo-2,3-dihydro-1H-benzimidazol-5-yl)-1-methyl-1H-pyrrole-2-carbonitrile: A novel, highly potent, selective, and orally active non-steroidal progesterone receptor agonist.

Raymond J. Unwalla, R. Winneker, E. Trybulski, 2007, Bioorganic & medicinal chemistry.

7-aryl 1,5-dihydro-benzo[e][1,4]oxazepin-2-ones and analogs as non-steroidal progesterone receptor antagonists.

R. Winneker, J. Wrobel, T. Berrodin, 2008, Bioorganic & medicinal chemistry.

Synthesis and progesterone receptor antagonist activities of 6-aryl benzimidazolones and benzothiazolones.

Z. Zhang, P. Zhang, Eugene A. Terefenko, 2001, Bioorganic & medicinal chemistry letters.

1-Methyl-1H-pyrrole-2-carbonitrile containing tetrahydronaphthalene derivatives as non-steroidal progesterone receptor antagonists.

R. Winneker, E. Trybulski, T. Berrodin, 2010, Bioorganic & medicinal chemistry letters.

5-Aryl indanones and derivatives as non-steroidal progesterone receptor modulators.

R. Winneker, E. Trybulski, T. Berrodin, 2009, Bioorganic & medicinal chemistry letters.

1,5-Dihydro-benzo[e][1,4]oxazepin-2(1H)-ones containing a 7-(5'-cyanopyrrol-2-yl) group as nonsteroidal progesterone receptor modulators.

Raymond J. Unwalla, R. Winneker, J. Wrobel, 2008, Bioorganic & medicinal chemistry letters.

1- or 3-(3-Amino-2-hydroxy-1-phenyl propyl)-1,3-dihydro-2H-benzimidazol-2-ones: potent, selective, and orally efficacious norepinephrine reuptake inhibitors.

D. Deecher, P. Mahaney, E. Trybulski, 2009, Journal of medicinal chemistry.