Daisuke Wakasugi

发表

A novel synthesis of bicyclo[3.3.0]oct-1-en-3-ones from cyclobutanones through [chloro(p-tolylsulfinyl)methylidene]cyclobutanes with ring expansion

T. Satoh, T. Kawashima, Hiroaki Kashima, 2005 .

A novel synthesis, including asymmetric synthesis, of 2,4,4-trisubstituted 2-cyclopentenones based on the reaction of 1-chlorovinyl p-tolyl sulfoxides with acetonitrile and its homologues

T. Satoh, Daisuke Wakasugi, 2005 .

A novel synthesis of 2,4,4-trisubstituted 2-cyclopentenones by consecutive reaction of 1-chlorovinyl p-tolyl sulfoxides with acetonitrile and its homologues

T. Satoh, Daisuke Wakasugi, 2003 .

A versatile synthesis, including asymmetric synthesis, of bicyclo[n.1.0]alkanes from cyclic ketones via the magnesium carbenoid 1,3-CH insertion as a key reaction

T. Satoh, Daisuke Wakasugi, S. Ogata, 2006 .

A method for synthesis of bicyclo [3.3.0 ]oct -1 -en -3 -ones from cyclobutanones with one-carbon ring expansion and its application to a formal synthesis of racemic 1-desoxyhypnophilin

T. Satoh, T. Kawashima, Hiroaki Kashima, 2007 .

A synthesis of bicyclo[n.1.0]alkanes having tert-butyl carboxylate or acetamide moiety via the intramolecular 1,3-CH insertion of magnesium carbenoids

T. Satoh, H. Saitoh, Daisuke Wakasugi, 2008 .

Design and synthesis of disubstituted (4-piperidinyl)-piperazine derivatives as potent acetyl-CoA carboxylase inhibitors.

F. Io, Hiroko Koretsune, D. Yamamoto, 2010, Bioorganic & medicinal chemistry letters.

Isoquinoline derivatives as potent CRTH2 antagonists: design, synthesis and SAR.

Kazuhito Watanabe, Susumu Yamanobe, Y. Sekiguchi, 2013, Bioorganic & medicinal chemistry.

Isoquinoline derivatives as potent CRTH2 receptor antagonists: synthesis and SAR.

Kazuhito Watanabe, Y. Sekiguchi, T. Koami, 2012, Bioorganic & medicinal chemistry letters.

Discovery of novel (4-piperidinyl)-piperazines as potent and orally active acetyl-CoA carboxylase 1/2 non-selective inhibitors: F-Boc and triF-Boc groups are acid-stable bioisosteres for the Boc group.

F. Io, Hiroko Koretsune, D. Yamamoto, 2011, Bioorganic & medicinal chemistry.

(4-Piperidinyl)-piperazine: a new platform for acetyl-CoA carboxylase inhibitors.

F. Io, Hiroko Koretsune, D. Yamamoto, 2009, Bioorganic & medicinal chemistry letters.

Lead identification of novel tetrahydroimidazo[1,2-a]pyridine-5-carboxylic acid derivative as a potent heparanase-1 inhibitor.

Sayaka Kato, H. Kakinuma, Sota Kato, 2022, Bioorganic & medicinal chemistry letters.

Isoquinoline derivatives as potent, selective, and orally active CRTH2 antagonists.

Kazuhito Watanabe, Y. Sekiguchi, Tetsuo Takayama, 2014, Chemical & pharmaceutical bulletin.

Structure-based lead optimization to improve potency and selectivity of a novel tetrahydroimidazo[1,2-a]pyridine-5-carboxylic acid series of heparanase-1 inhibitor.

H. Kakinuma, H. Miyagawa, Mayumi Endo, 2023, Bioorganic & medicinal chemistry.

Design and synthesis of disubstituted (4-piperidinyl)-piperazine derivatives as potent acetyl-CoA carboxylase inhibitors.

Hiroko Koretsune, D. Yamamoto, Akira Hiratate, 2010, Bioorganic & medicinal chemistry letters.

(4-Piperidinyl)-piperazine: a new platform for acetyl-CoA carboxylase inhibitors.

Hiroko Koretsune, D. Yamamoto, Akira Hiratate, 2009, Bioorganic & medicinal chemistry letters.