Yingjun Li

发表

2,4-Diarylamino-pyrimidines as kinase inhibitors co-targeting IGF1R and EGFR(L⁸⁵⁸R/T⁷⁹⁰M).

J. Smaill, Jian Ding, Lin-jiang Tong, 2015, Bioorganic & medicinal chemistry letters.

Design, synthesis, and biological evaluation of 3-(1H-1,2,3-triazol-1-yl)benzamide derivatives as Potent Pan Bcr-Abl inhibitors including the threonine(315)→isoleucine(315) mutant.

Xiaoyun Lu, Zheng-chao Tu, Fengxiang Zhang, 2012, Journal of medicinal chemistry.

N-(3-Ethynyl-2,4-difluorophenyl)sulfonamide Derivatives as Selective Raf Inhibitors.

Yong Xu, J. Smaill, Donghai Wu, 2015, ACS medicinal chemistry letters.

Synthesis and biological evaluation of novel thiadiazole amides as potent Cdc25B and PTP1B inhibitors.

Kun Jin, Jia Li, Li-xin Gao, 2014, Bioorganic & medicinal chemistry letters.

Design and Synthesis of Tetrazole- and Pyridine-Containing Itraconazole Analogs as Potent Angiogenesis Inhibitors.

Jun O. Liu, K. Pasunooti, W. Shi, 2020, ACS medicinal chemistry letters.

Pyrazole-4-Carboxamide (YW2065): A Therapeutic Candidate for Colorectal Cancer via Dual Activities of Wnt/β-Catenin Signaling Inhibition and AMP-Activated Protein Kinase (AMPK) Activation.

M. Xia, S. Sakamuru, Hong Yang, 2019, Journal of medicinal chemistry.

Evaluation of Benzamide Derivatives as New Influenza A Nucleoprotein Inhibitors

Yanmei Zhang, Zheng-chao Tu, M. Tortorella, 2016 .

Determination of A Novel Selective B-RafV600E Inhibitor (LXK4) in Dog Plasma by HPLC–MS/MS and its Application in a Pharmacokinetic Study

R. Dai, Jifeng Deng, Huimin Cheng, 2016, Chromatographia.

Triazole-Based Inhibitors of the Wnt/β-Catenin Signaling Pathway Improve Glucose and Lipid Metabolisms in Diet-Induced Obese Mice.

M. Xia, S. Sakamuru, Hong Yang, 2019, Journal of medicinal chemistry.

Discovery of a potent GLUT inhibitor using rapafucin 3D microarrays.

Jun O. Liu, S. Sukumar, J. Locasale, 2019, Angewandte Chemie.

Novel Tetrazole-Containing Analogues of Itraconazole as Potent Antiangiogenic Agents with Reduced Cytochrome P450 3A4 Inhibition.

Jun O. Liu, K. Pasunooti, W. Shi, 2018, Journal of medicinal chemistry.

Discovery of BRAF/HDAC Dual Inhibitors Suppressing Proliferation of Human Colorectal Cancer Cells

Ruxi Qi, Zheng-chao Tu, Zhang Zhang, 2022, Frontiers in Chemistry.

Structure Based Design of N-(3-((1H-Pyrazolo[3,4-b]pyridin-5-yl)ethynyl)benzenesulfonamides as Selective Leucine-Zipper and Sterile-α Motif Kinase (ZAK) Inhibitors.

Yan Zhang, Yong Xu, Chih-Yang Huang, 2017, Journal of medicinal chemistry.

Structure-activity study on a series of α-glutamic acid scaffold based compounds as new ADAMTS inhibitors.

Honglin Li, Xiaofeng Liu, Lei Duan, 2011, Bioorganic & Medicinal Chemistry Letters.

Discovery of a Potent GLUT Inhibitor from a Library of Rapafucins by Using 3D Microarrays

Jun O. Liu, S. Sukumar, J. Locasale, 2019, Angewandte Chemie.

Structure Based Design of N-(3-((1H-Pyrazolo[3,4-b]pyridin-5-yl)ethynyl)benzenesulfonamides as Selective Leucine-Zipper and Sterile-α Motif Kinase (ZAK) Inhibitors.

Yan Zhang, Yong Xu, Chih-Yang Huang, 2017, Journal of medicinal chemistry.