M. Charest

A Convergent Enantioselective Route to Structurally Diverse 6-Deoxytetracycline Antibiotics

Andrew G Myers, C. Lerner, D. Siegel, 2005, Science.

Synthesis of (-)-tetracycline.

D. Siegel, A. Myers, M. Charest, 2005, Journal of the American Chemical Society.

Synthesis of a broad array of highly functionalized, enantiomerically pure cyclohexanecarboxylic acid derivatives by microbial dihydroxylation of benzoic acid and subsequent oxidative and rearrangement reactions.

D. Siegel, A. Myers, D. Buzard, 2001, Organic letters.

A robust platform for the synthesis of new tetracycline antibiotics.

C. Lerner, D. Siegel, P. Wright, 2008, Journal of the American Chemical Society.

Design and synthesis of highly potent HIV protease inhibitors with activity against resistant virus.

W. Schleif, L. Gabryelski, E. Emini, 2003, Bioorganic & medicinal chemistry letters.